SCHEMBL7449277

SCHEMBL7449277

CCCc1ccccc1C(=O)NNC(=O)c1csc(-c2ccccc2OCc2ccccc2)n1

nearest known ligand 0.47

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PTGER1 P34995 6/20 0.47
TLR7 Q9NYK1 9/20 0.45
NPC1 O15118 1/20 0.43
PTGER4 P35408 4/20 0.43
PTGER3 P43115 4/20 0.43
PTGER2 P43116 4/20 0.43
OPRK1 P41145 1/20 0.42
KMT2A Q03164 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7449236 0.94 PTGER1 (0.46) PTGER1TLR7NPC1PTGER4PTGER3
SCHEMBL7446264 0.93 TLR7 (0.50) PTGER1TLR7NPC1PTGER4PTGER3
SCHEMBL7449102 0.88 PTGER1 (0.46) PTGER1TLR7PTGER4PTGER3PTGER2
SCHEMBL7448360 0.86 TLR7 (0.50) PTGER1TLR7NPC1KMT2A
SCHEMBL7448167 0.86 PTGER1 (0.50) PTGER1TLR7NPC1
SCHEMBL7448062 0.85 TLR7 (0.48) PTGER1TLR7NPC1
SCHEMBL7549322 0.83 PTGER1 (0.49) PTGER1TLR7NPC1
SCHEMBL7447138 0.82 PTGER1 (0.54) PTGER1TLR7
SCHEMBL7512520 0.82 PTGER1 (0.42) PTGER1TLR7PTGER4PTGER3PTGER2
SCHEMBL7449446 0.82 PTGER1 (0.45) PTGER1TLR7PTGER4PTGER3PTGER2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0977743-A1 PROTEASE INHIBITORS Smithkline Beecham (US) 2000-02-09 EP claimed
WO-1998049152-A1 PROTEASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 1998-11-05 WO claimed
EP-0977743-A1 PROTEASE INHIBITORS Smithkline Beecham (US) 2000-02-09 EP disclosed
WO-1998049152-A1 PROTEASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 1998-11-05 WO disclosed