SCHEMBL7449404

SCHEMBL7449404

Nc1ccc(-c2ccccc2)c(SC(F)(F)F)c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX5AP P20292 1/20 0.42
FEN1 P39748 1/20 0.42
ALDH1A1 P00352 5/20 0.41
TDP1 Q9NUW8 3/20 0.41
KDM4E B2RXH2 2/20 0.41
TSHR P16473 3/20 0.40
GLA P06280 2/20 0.40
GAA P10253 2/20 0.40
POLB P06746 2/20 0.40
MAOA P21397 1/20 0.38
PDK2 Q15119 3/20 0.38
HSD17B10 Q99714 2/20 0.38
CYP3A4 P08684 2/20 0.38
TAAR1 Q96RJ0 1/20 0.38
NPC1 O15118 3/20 0.36
PTGDR2 Q9Y5Y4 1/20 0.36
SMN1; SMN2 Q16637 3/20 0.35
MAPK1 P28482 2/20 0.35
RAB9A P51151 2/20 0.35
TP53 P04637 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6902556 0.80 MAOA (0.45) ALDH1A1TDP1KDM4ETSHRGLA
SCHEMBL6282287 0.79 ALOX5AP (0.50) ALOX5APFEN1ALDH1A1TDP1KDM4E
SCHEMBL5175215 0.77 ALOX5AP (0.44) ALOX5APFEN1ALDH1A1KDM4EHSD17B10
SCHEMBL3781939 0.77 MAOA (0.42) ALOX5APFEN1ALDH1A1TDP1KDM4E
SCHEMBL28327988 0.76 PDK2 (0.43) ALDH1A1TDP1TSHRPDK2SMN1; SMN2
SCHEMBL3789390 0.75 ALDH1A1 (0.51) ALDH1A1TDP1KDM4ETSHRGLA
SCHEMBL4250948 0.74 ALDH1A1 (0.41) ALOX5APFEN1ALDH1A1TDP1KDM4E
SCHEMBL1926441 0.73 TSHR (0.70) ALDH1A1TDP1TSHRGLAGAA
SCHEMBL3805104 0.72 ADORA2A (0.41) ALDH1A1TDP1KDM4ETSHRGLA
SCHEMBL9404028 0.72 KDM4E (0.48) ALOX5APFEN1ALDH1A1TDP1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0946528-A2 OXYGEN OR SULFUR CONTAINING 5-MEMBERED HETEROAROMATICS AS FACTOR Xa INHIBITORS Du Pont Pharmaceuticals Company (US) 1999-10-06 EP disclosed
WO-1998028282-A2 OXYGEN OR SULFUR CONTAINING 5-MEMBERED HETEROAROMATICS AS FACTOR Xa INHIBITORS DU PONT PHARMACEUTICALS COMPANY (US) 1998-07-02 WO disclosed