SCHEMBL7449552

SCHEMBL7449552

CCOc1cc2c(cc1OCC)C(=O)C(NC(=O)C(F)(F)F)CC2

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.57
ACHE P22303 1/20 0.46
HTT P42858 1/20 0.43
NCOA1 Q15788 1/20 0.43
NCOA3 Q9Y6Q9 1/20 0.43
LMNA P02545 2/20 0.38
GAA P10253 1/20 0.38
POLB P06746 1/20 0.37
MAPT P10636 1/20 0.37
NQO2 P16083 5/20 0.35
MTNR1A P48039 5/20 0.35
MTNR1B P49286 5/20 0.35
ALDH1A1 P00352 1/20 0.35
NPC1 O15118 1/20 0.35
RAB9A P51151 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
SSTR4 P31391 1/20 0.34
KMT2A Q03164 1/20 0.34
PDE4A P27815 1/20 0.34
PDE4B Q07343 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21798820 0.87 HTT (0.57) KDM4EACHEHTTNCOA1NCOA3
SCHEMBL7027773 0.81 HTT (0.51) KDM4EHTTNCOA1NCOA3LMNA
SCHEMBL5889352 0.81 HTT (0.51) KDM4EHTTNCOA1NCOA3LMNA
SCHEMBL8063041 0.81 HTT (0.51) KDM4EHTTNCOA1NCOA3LMNA
SCHEMBL8075935 0.77 RAB9A (0.39) KDM4EHTTNCOA1NCOA3LMNA
SCHEMBL8075930 0.77 RAB9A (0.39) KDM4EHTTNCOA1NCOA3LMNA
SCHEMBL8070827 0.74 HTT (0.51) KDM4EHTTNCOA1NCOA3LMNA
SCHEMBL7248408 0.74 KDM4E (0.49) KDM4EACHEHTTNCOA1NCOA3
SCHEMBL8070825 0.74 HTT (0.51) KDM4EHTTNCOA1NCOA3LMNA
SCHEMBL7568637 0.74 KDM4E (0.49) KDM4EACHEHTTNCOA1NCOA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2002000609-A2 2,6,7-SUBSTITUTED TETRALINES USEFUL FOR THE PREPARATION OF MEDICAMENTS WITH PHOSPHODIESTERASE IV INHIBITORY ACTIVITY SIGMA-TAU INDUSTRIE FARMACEUTICHE RIUNITE S.P.A. (IT) 2002-01-03 WO claimed
WO-2002000609-A2 2,6,7-SUBSTITUTED TETRALINES USEFUL FOR THE PREPARATION OF MEDICAMENTS WITH PHOSPHODIESTERASE IV INHIBITORY ACTIVITY SIGMA-TAU INDUSTRIE FARMACEUTICHE RIUNITE S.P.A. (IT) 2002-01-03 WO disclosed