SCHEMBL7449941

SCHEMBL7449941

COc1ccc(COC(=O)C2CCCN2Cc2ccc(OC)cc2)cc1

nearest known ligand 0.56

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.56
ALDH1A1 P00352 3/20 0.54
SPHK2 Q9NRA0 1/20 0.52
POLB P06746 1/20 0.52
HRH3 Q9Y5N1 1/20 0.50
OPRM1 P35372 1/20 0.49
OPRK1 P41145 1/20 0.49
SPHK1 Q9NYA1 1/20 0.49
TSHR P16473 1/20 0.48
SCN3A Q9NY46 1/20 0.47
MEN1 O00255 1/20 0.47
KMT2A Q03164 1/20 0.47
GAA P10253 1/20 0.47
HPGD P15428 1/20 0.47
FKBP1A P62942 1/20 0.47
MAOA P21397 1/20 0.47
MAOB P27338 1/20 0.47
LTA4H P09960 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21869793 0.95 POLB (0.58) KDM4EALDH1A1SPHK2POLBSPHK1
SCHEMBL7625352 0.86 KDM4E (0.73) KDM4EALDH1A1POLBHRH3TSHR
SCHEMBL9650151 0.85 KDM4E (0.56) KDM4EALDH1A1SPHK2POLBHRH3
SCHEMBL21409037 0.84 SMN1; SMN2 (0.56) KDM4ESPHK2HRH3OPRM1OPRK1
SCHEMBL10349406 0.84 KDM4E (0.57) KDM4EALDH1A1HRH3OPRM1OPRK1
SCHEMBL2274909 0.84 POLB (0.61) KDM4EALDH1A1POLBSPHK1MEN1
SCHEMBL2274911 0.84 POLB (0.61) KDM4EALDH1A1POLBSPHK1MEN1
SCHEMBL28957118 0.82 FKBP1A (0.58) ALDH1A1FKBP1A
SCHEMBL7458698 0.81 MCHR1 (0.53) KDM4EALDH1A1POLBHRH3
SCHEMBL6228519 0.80 CYP3A4 (0.55) KDM4EOPRM1OPRK1GAAHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1137412-A4 SUBSTITUTED NITROGEN HETEROCYCLIC COMPOUNDS AND THERAPEUTIC USES THEREOF AMERICAN BIOGENETIC SCIENCES (US) 2002-04-03 EP disclosed
EP-1137412-A2 SUBSTITUTED NITROGEN HETEROCYCLIC COMPOUNDS AND THERAPEUTIC USES THEREOF AMERICAN BIOGENETIC SCIENCES, INC. (US) 2001-10-04 EP disclosed
WO-2000033788-A2 SUBSTITUTED NITROGEN HETEROCYCLIC COMPOUNDS AND THERAPEUTIC USES THEREOF AMERICAN BIOGENETIC SCIENCES INC. (US) 2000-06-15 WO disclosed