SCHEMBL7450220

SCHEMBL7450220

BrN(c1ccccc1)c1nccc(-c2ccncc2)n1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GABRA1 P14867 1/20 0.43
GABRG2 P18507 1/20 0.43
GABRB3 P28472 1/20 0.43
GABRA5 P31644 1/20 0.43
GABRA3 P34903 1/20 0.43
AURKA O14965 1/20 0.42
HSP90AA1 P07900 1/20 0.42
PRKACA P17612 1/20 0.42
ADORA2A P29274 1/20 0.42
NPC1 O15118 3/20 0.41
AR P10275 2/20 0.41
CYP1A2 P05177 2/20 0.41
CYP3A4 P08684 2/20 0.41
CYP2D6 P10635 2/20 0.41
CYP2C9 P11712 2/20 0.41
CYP2C19 P33261 2/20 0.41
RAB9A P51151 2/20 0.41
NOTUM Q6P988 1/20 0.39
KMT2A Q03164 2/20 0.39
KDM4E B2RXH2 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10973799 0.81 GSK3B (0.51) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL7454799 0.77 MAPT (0.46) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL7470679 0.75 HIF1A (0.41) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL12073354 0.74 AURKA (0.53) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL18905473 0.72 GABRA1 (0.71) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL10918699 0.72 DYRK1A (0.53) NPC1ARCYP1A2CYP3A4CYP2D6
SCHEMBL10973666 0.71 GSK3B (0.55) AURKAHSP90AA1PRKACAADORA2ANPC1
SCHEMBL7445002 0.71 CYP2D6 (0.44) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL22377088 0.69 GABRA1 (0.68) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL28886710 0.68 AURKA (0.55) AURKAHSP90AA1PRKACAADORA2ARAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1115721-A1 PYRIMIDONE DERIVATIVES MITSUBISHI CHEMICAL CORPORATION (JP) 2001-07-18 EP disclosed
WO-2000018758-A1 PYRIMIDONE DERIVATIVES MITSUBISHI CHEMICAL CORPORATION (JP) 2000-04-06 WO disclosed