SCHEMBL7445002

SCHEMBL7445002

CCCCON(c1ccccc1)c1nccc(-c2ccncc2)n1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 4/20 0.44
CYP3A4 P08684 1/20 0.44
CYP19A1 P11511 2/20 0.41
CYP2C9 P11712 2/20 0.41
CYP2C19 P33261 2/20 0.41
CYP1A2 P05177 1/20 0.41
NPC1 O15118 3/20 0.40
MAPT P10636 5/20 0.39
KDM4E B2RXH2 3/20 0.39
L3MBTL1 Q9Y468 2/20 0.39
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
ALDH1A1 P00352 2/20 0.39
RAB9A P51151 2/20 0.39
LMNA P02545 1/20 0.39
TSHR P16473 1/20 0.39
HSD17B10 Q99714 1/20 0.39
ATP4A P20648 7/20 0.38
ATP4B P51164 7/20 0.38
HPGD P15428 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5400033 0.76 GSK3B (0.52) SMN1; SMN2
SCHEMBL7454799 0.76 MAPT (0.46) CYP2D6CYP3A4CYP2C9CYP2C19CYP1A2
SCHEMBL10973799 0.74 GSK3B (0.51) CYP2D6CYP3A4CYP2C9CYP2C19CYP1A2
SCHEMBL5400026 0.71 GCGR (0.42) CYP2D6CYP3A4GCGR
SCHEMBL7450220 0.71 GABRA1 (0.43) CYP2D6CYP3A4CYP19A1CYP2C9CYP2C19
SCHEMBL12073354 0.68 AURKA (0.53) MAPTKDM4EL3MBTL1MEN1KMT2A
SCHEMBL28194680 0.68 ALDH1A1 (0.47) CYP3A4NPC1MAPTKDM4EALDH1A1
SCHEMBL27361074 0.68 ALDH1A1 (0.47) CYP3A4NPC1MAPTKDM4EALDH1A1
SCHEMBL10918699 0.66 DYRK1A (0.53) CYP2D6CYP3A4CYP2C9CYP2C19CYP1A2
SCHEMBL7470679 0.66 HIF1A (0.41) CYP2D6CYP3A4CYP2C9CYP2C19CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1115721-A1 PYRIMIDONE DERIVATIVES MITSUBISHI CHEMICAL CORPORATION (JP) 2001-07-18 EP disclosed
WO-2000018758-A1 PYRIMIDONE DERIVATIVES MITSUBISHI CHEMICAL CORPORATION (JP) 2000-04-06 WO disclosed