SCHEMBL7450424

SCHEMBL7450424

O=C(c1ccc(OCCCN2CCCC2)cc1)c1ccsc1

nearest known ligand 0.67

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 5/20 0.67
ALDH1A1 P00352 3/20 0.66
PSMB1 P20618 1/20 0.65
PSMB5 P28074 1/20 0.65
PSMB2 P49721 1/20 0.65
HRH4 Q9H3N8 1/20 0.64
LTA4H P09960 1/20 0.61
HRH3 Q9Y5N1 7/20 0.60
MAOB P27338 1/20 0.57
GCGR P47871 1/20 0.57
BCHE P06276 1/20 0.56
ACHE P22303 1/20 0.56
SMN1; SMN2 Q16637 1/20 0.54
CACNA1B Q00975 1/20 0.54
POLB P06746 1/20 0.53
MAPT P10636 1/20 0.53
KCNH2 Q12809 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8337044 0.99 KDM4E (0.68) KDM4EALDH1A1PSMB1PSMB5PSMB2
SCHEMBL4543175 0.94 PSMB1 (0.75) KDM4EALDH1A1PSMB1PSMB5PSMB2
Water SCHEMBL8476776 0.93 PSMB1 (0.73) KDM4EALDH1A1PSMB1PSMB5PSMB2
SCHEMBL7443953 0.93 PSMB1 (0.78) KDM4EALDH1A1PSMB1PSMB5PSMB2
Hydrochloric Acid SCHEMBL8475814 0.93 PSMB1 (0.73) KDM4EALDH1A1PSMB1PSMB5PSMB2
Water SCHEMBL8476448 0.91 PSMB1 (0.76) KDM4EALDH1A1PSMB1PSMB5PSMB2
Hydrochloric Acid SCHEMBL7451065 0.91 PSMB1 (0.76) KDM4EALDH1A1PSMB1PSMB5PSMB2
SCHEMBL7447270 0.83 SMN1; SMN2 (0.61) KDM4EALDH1A1PSMB1PSMB5PSMB2
SCHEMBL8641421 0.82 PSMB1 (0.62) KDM4EALDH1A1PSMB1PSMB5PSMB2
SCHEMBL7441221 0.82 ESR1 (0.49) KDM4EALDH1A1PSMB1PSMB5PSMB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5948796-A OSTEOPOROSIS, CANCER, CARDIOVASCULAR DISORDERS ELI LILLY AND COMPANY (US) 1999-09-07 US disclosed
EP-0863755-A4 ANTITHROMBOTIC DIAMINES LILLY CO ELI (US) 1999-01-20 EP disclosed
EP-0863755-A1 ANTITHROMBOTIC DIAMINES ELI LILLY AND COMPANY (US) 1998-09-16 EP disclosed
WO-1997025033-A1 ANTITHROMBOTIC DIAMINES ELI LILLY AND COMPANY (US) 1997-07-17 WO disclosed