SCHEMBL7450448

SCHEMBL7450448

CC(C)CC(NC(=O)c1ccc(CN)cc1)C(=O)N(C)C#N

nearest known ligand 0.58

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CTSB P07858 9/20 0.58
CTSL P07711 9/20 0.53
CTSS P25774 5/20 0.53
CTSK P43235 5/20 0.53
TAS1R3 Q7RTX0 1/20 0.46
TAS1R1 Q7RTX1 1/20 0.46
CA2 P00918 2/20 0.44
CA1 P00915 1/20 0.44
HPGDS O60760 1/20 0.44
F3 P13726 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6203497 0.89 CTSB (0.55) CTSBCTSLCTSSCTSKF3
SCHEMBL6183809 0.88 CTSB (0.61) CTSBCTSLCTSSCTSKCA2
SCHEMBL6182874 0.88 CTSB (0.61) CTSBCTSLCTSSCTSKCA2
SCHEMBL6183805 0.88 CTSB (0.61) CTSBCTSLCTSSCTSKCA2
SCHEMBL6182791 0.88 CTSB (0.61) CTSBCTSLCTSSCTSKCA2
SCHEMBL7452244 0.85 CTSB (0.61) CTSBCTSLCTSSCTSK
SCHEMBL7511749 0.84 CA2 (0.67) CTSBCTSLCTSSCTSKCA2
SCHEMBL6180502 0.84 CTSB (0.56) CTSBCTSLCTSSCTSKCA2
SCHEMBL6183292 0.83 CTSB (0.58) CTSBCTSLCTSSCTSKTAS1R3
SCHEMBL5925030 0.83 CTSB (0.58) CTSBCTSLCTSSCTSKCA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1161415-A2 N-CYANOMETHYLAMIDES AS PROTEASE INHIBITORS AXYS PHARMACEUTICALS, INC. (US) 2001-12-12 EP disclosed
WO-2000055126-A2 N-CYANOMETHYLAMIDES AS PROTEASE INHIBITORS AXYS PHARMACEUTICALS, INC. (US) 2000-09-21 WO disclosed