SCHEMBL7450463

SCHEMBL7450463

C1=Cc2c(ccc3c2ccc2ccccc23)SN1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPRT1 P00492 4/20 0.47
ALDH1A1 P00352 5/20 0.40
HSD17B10 Q99714 3/20 0.40
TDP1 Q9NUW8 2/20 0.40
CYP2A6 P11509 1/20 0.40
TSHR P16473 1/20 0.40
PAX8 Q06710 1/20 0.36
HPGD P15428 3/20 0.36
CYP1A2 P05177 3/20 0.36
HIF1A Q16665 2/20 0.36
LMNA P02545 2/20 0.36
MAPK1 P28482 2/20 0.36
CYP2C9 P11712 2/20 0.36
CYP2C19 P33261 2/20 0.36
MEN1 O00255 1/20 0.36
USP2 O75604 1/20 0.36
TP53 P04637 1/20 0.36
CYP2D6 P10635 1/20 0.36
ALOX12 P18054 1/20 0.36
KMT2A Q03164 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3073175 0.91 ALDH1A1 (0.39) HPRT1ALDH1A1HSD17B10TDP1CYP2A6
Chrysene SCHEMBL29355502 0.68 HPRT1 (1.00) HPRT1ALDH1A1HSD17B10TDP1CYP2A6
Chrysene SCHEMBL29792076 0.68 HPRT1 (1.00) HPRT1ALDH1A1HSD17B10TDP1CYP2A6
SCHEMBL29451340 0.68 HPRT1 (1.00) HPRT1ALDH1A1HSD17B10TDP1CYP2A6
SCHEMBL25510 0.68 HPRT1 (1.00) HPRT1ALDH1A1HSD17B10TDP1CYP2A6
Chrysene SCHEMBL384031 0.68 HPRT1 (1.00) HPRT1ALDH1A1HSD17B10TDP1CYP2A6
Chrysene SCHEMBL9786466 0.68 HPRT1 (1.00) HPRT1ALDH1A1HSD17B10TDP1CYP2A6
SCHEMBL31177955 0.68 HPRT1 (1.00) HPRT1ALDH1A1HSD17B10TDP1CYP2A6
Chrysene SCHEMBL27115 0.68 HPRT1 (1.00) HPRT1ALDH1A1HSD17B10TDP1CYP2A6
SCHEMBL29640482 0.68 HPRT1 (1.00) HPRT1ALDH1A1HSD17B10TDP1CYP2A6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117263999-A Camptothecin prodrugs and pharmaceutical compositions thereof 天津和美奥康医药科技有限公司 2023-12-22 CN disclosed
EP-1261594-A1 5,10-DIHYDROACRIDINES AS CALCIUM CHANNEL BLOCKERS Neuromed Technologies, Inc. (CA) 2002-12-04 EP disclosed
US-6310059-B1 CONSTRAINED FUSED RING DERIVATIVES OF PIPERIDINE OR PIPERAZINE LINKED TO HYDROPHOBIC SUBSTITUENTS WHICH ENHANCE CALCIUM CHANNEL BLOCKING ACTIVITY; COMBINATORIAL LIBRARIES FOR DRUG SCREENING NEUROMED TECHNOLOGIES, INC. (CA) 2001-10-30 US disclosed
WO-2001049670-A1 5,10-DIHYDROACRIDINES AS CALCIUM CHANNEL BLOCKERS NEUROMED TECHNOLOGIES, INC. (CA) 2001-07-12 WO disclosed