SCHEMBL7450648

SCHEMBL7450648

[C]1=C(c2nc3ccccc3o2)Cc2ccccc2O1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 6/20 0.42
ALDH1A1 P00352 6/20 0.42
RAB9A P51151 5/20 0.42
HSD17B10 Q99714 5/20 0.42
HPGD P15428 5/20 0.42
TP53 P04637 4/20 0.42
KDM4E B2RXH2 4/20 0.42
MEN1 O00255 3/20 0.42
KMT2A Q03164 3/20 0.42
SMN1; SMN2 Q16637 3/20 0.42
MAPT P10636 3/20 0.42
PKM P14618 2/20 0.42
HCRTR1 O43613 1/20 0.42
CYP1A2 P05177 1/20 0.42
CYP2C9 P11712 1/20 0.42
CYP2C19 P33261 1/20 0.42
ATM Q13315 1/20 0.41
ALOX5 P09917 1/20 0.41
CHRM2 P08172 1/20 0.38
CHRM4 P08173 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7657314 0.72 MAOB (0.43) NPC1ALDH1A1RAB9AHSD17B10HPGD
SCHEMBL29531707 0.72 NPC1 (0.69) NPC1ALDH1A1RAB9AHSD17B10HPGD
SCHEMBL824375 0.72 NPC1 (0.69) NPC1ALDH1A1RAB9AHSD17B10HPGD
SCHEMBL482462 0.70 KDM4E (0.34) NPC1ALDH1A1RAB9AHSD17B10HPGD
SCHEMBL4747222 0.69 MAOA (0.39) TP53
SCHEMBL2140405 0.69 ALDH1A1 (0.49) NPC1ALDH1A1RAB9AHSD17B10HPGD
SCHEMBL31170 0.65 NPC1 (0.81) NPC1ALDH1A1RAB9AHSD17B10HPGD
SCHEMBL171055 0.65 TOP2A (0.62) NPC1ALDH1A1RAB9AHSD17B10HPGD
SCHEMBL21674121 0.65 NPC1 (0.63) NPC1ALDH1A1RAB9AHSD17B10HPGD
SCHEMBL29504749 0.65 TOP2A (0.62) NPC1ALDH1A1RAB9AHSD17B10HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2001074793-A2 SUBSTITUTED THIAZOLES AND THE USE THEREOF AS INHIBITORS OF PLASMINOGEN ACTIVATOR INHIBITOR-1 3-DIMENSIONAL PHARMACEUTICALS, INC. (US) 2001-10-11 WO disclosed