SCHEMBL7450674

SCHEMBL7450674

CC(=O)N[C@@H](C(=O)O)c1ccc(OC(C)=O)cc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 3/20 0.51
GAA P10253 2/20 0.51
ALDH1A1 P00352 1/20 0.51
HSP90AA1 P07900 1/20 0.51
LMNA P02545 3/20 0.47
ELANE P08246 1/20 0.46
HSD17B10 Q99714 1/20 0.45
ACACB O00763 4/20 0.43
ACACA Q13085 3/20 0.43
KDM4E B2RXH2 2/20 0.43
CYP3A4 P08684 2/20 0.43
POLB P06746 1/20 0.43
PKM P14618 1/20 0.43
ABCB11 O95342 1/20 0.43
ESR1 P03372 1/20 0.43
ADRA2A P08913 1/20 0.43
CYP2C9 P11712 1/20 0.43
TSHR P16473 1/20 0.43
PDE4A P27815 1/20 0.43
ADRA1A P35348 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11698235 1.00 MAPT (0.51) MAPTGAAALDH1A1HSP90AA1LMNA
SCHEMBL29401218 1.00 MAPT (0.51) MAPTGAAALDH1A1HSP90AA1LMNA
Valine SCHEMBL11699886 0.89 MAPT (0.42) MAPTGAAALDH1A1HSP90AA1LMNA
SCHEMBL11697241 0.85 ATM (0.56) ALDH1A1ACACBACACACYP3A4TSHR
SCHEMBL11349043 0.82 CTSS (0.51) MAPTGAAALDH1A1HSP90AA1LMNA
SCHEMBL6965264 0.79 ACACB (0.60) ACACBACACA
SCHEMBL11693549 0.79 FOLH1 (0.56) MAPTALDH1A1CYP3A4ESR1TSHR
SCHEMBL3376625 0.78 SRC (0.52) ALDH1A1LMNAPOLBKMT2AATM
SCHEMBL627377 0.78 SRC (0.52) ALDH1A1LMNAPOLBKMT2AATM
SCHEMBL4250144 0.78 SRC (0.52) ALDH1A1LMNAPOLBKMT2AATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0918768-B1 AROMATIC AMIDINE DERIVATIVES USEFUL AS SELECTIVE THROMBIN INHIBITORS C & C RES LAB (KR) 2002-01-09 EP disclosed
US-6201006-B1 ANTICOAGULANTS C & C RESEARCH LABORATORIES (KR) 2001-03-13 US disclosed
EP-0918768-A1 AROMATIC AMIDINE DERIVATIVES USEFUL AS SELECTIVE THROMBIN INHIBITORS C & C Research Laboratories (KR) 1999-06-02 EP disclosed
WO-1997045424-A1 AROMATIC AMIDINE DERIVATIVES USEFUL AS SELECTIVE THROMBIN INHIBITORS C & C RESEARCH LABORATORIES (KR) 1997-12-04 WO disclosed