SCHEMBL7450747

SCHEMBL7450747

O=C(Nc1ccnc(Cl)c1)c1nnn2c1CS(=O)(=O)c1cc(Cl)ccc1-2

nearest known ligand 0.61

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 3/20 0.61
SMARCA2 P51531 5/20 0.38
SMARCA4 P51532 4/20 0.38
CNR1 P21554 2/20 0.36
CNR2 P34972 1/20 0.36
GRM4 Q14833 2/20 0.35
GRM1 Q13255 1/20 0.35
THRB P10828 1/20 0.35
SMURF1 Q9HCE7 1/20 0.34
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12067838 0.92 GRM5 (0.59) GRM5SMARCA2SMARCA4CNR1CNR2
SCHEMBL12065522 0.90 GRM5 (0.62) GRM5SMARCA2SMARCA4GRM4GRM1
SCHEMBL7452726 0.89 GRM5 (0.58) GRM5SMARCA2SMARCA4THRBNPC1
SCHEMBL12067836 0.81 GRM5 (0.52) GRM5SMARCA2SMARCA4CNR1CNR2
SCHEMBL7459153 0.80 GRM5 (0.72) GRM5SMARCA2SMARCA4CNR1CNR2
SCHEMBL7453851 0.78 GRM5 (0.69) GRM5SMARCA2SMARCA4CNR1CNR2
SCHEMBL7445410 0.76 GRM5 (1.00) GRM5SMARCA2SMARCA4NPC1RAB9A
SCHEMBL7454651 0.75 GRM5 (0.52) GRM5SMARCA2SMARCA4CNR1CNR2
SCHEMBL7454592 0.73 GRM5 (0.68) GRM5SMARCA2SMARCA4GRM4NPC1
SCHEMBL7453211 0.73 GRM5 (0.55) GRM5SMARCA2SMARCA4GRM4SMURF1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011151361-A1 NOVEL COMPOUNDS GLAXO GROUP LIMITED (GB) 2011-12-08 WO disclosed
WO-2011151361-A1 NOVEL COMPOUNDS GLAXO GROUP LIMITED (GB) 2011-12-08 WO disclosed