SCHEMBL7450866

SCHEMBL7450866

CCN(CC)c1ccc(C(=O)NC(CC(C)C)C(=O)N(C)C#N)cc1

nearest known ligand 0.57

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CTSB P07858 11/20 0.57
CTSL P07711 12/20 0.52
CTSS P25774 7/20 0.52
CTSK P43235 7/20 0.52
CNR2 P34972 1/20 0.45
TAS1R3 Q7RTX0 2/20 0.43
TAS1R1 Q7RTX1 2/20 0.43
CTSF Q9UBX1 1/20 0.42
CA12 O43570 1/20 0.42
CA1 P00915 1/20 0.42
CA9 Q16790 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7507894 0.90 CTSB (0.46) CTSBCTSLCTSSCTSKCNR2
SCHEMBL7452244 0.89 CTSB (0.61) CTSBCTSLCTSSCTSKCTSF
SCHEMBL6182114 0.85 CTSB (0.58) CTSBCTSLCTSSCTSKCTSF
SCHEMBL6183809 0.84 CTSB (0.61) CTSBCTSLCTSSCTSKCTSF
SCHEMBL6183805 0.84 CTSB (0.61) CTSBCTSLCTSSCTSKCTSF
SCHEMBL6182791 0.84 CTSB (0.61) CTSBCTSLCTSSCTSKCTSF
SCHEMBL6182874 0.84 CTSB (0.61) CTSBCTSLCTSSCTSKCTSF
SCHEMBL6180502 0.83 CTSB (0.56) CTSBCTSLCTSSCTSKCTSF
SCHEMBL6181880 0.83 CTSB (0.56) CTSBCTSLCTSSCTSKCTSF
SCHEMBL7450448 0.82 CTSB (0.58) CTSBCTSLCTSSCTSKTAS1R3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1161415-A2 N-CYANOMETHYLAMIDES AS PROTEASE INHIBITORS AXYS PHARMACEUTICALS, INC. (US) 2001-12-12 EP disclosed
WO-2000055126-A2 N-CYANOMETHYLAMIDES AS PROTEASE INHIBITORS AXYS PHARMACEUTICALS, INC. (US) 2000-09-21 WO disclosed