SCHEMBL7452011

SCHEMBL7452011

O=C(c1ccc(OCCN2CCCC2)cc1)c1c(-c2ccc(OCCN3CCCC3)cc2)oc2ccccc12

nearest known ligand 0.64

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 7/20 0.64
BCHE P06276 5/20 0.64
CNR2 P34972 4/20 0.64
ACHE P22303 2/20 0.64
LTA4H P09960 1/20 0.62
L3MBTL1 Q9Y468 1/20 0.60
PSMB1 P20618 1/20 0.59
PSMB5 P28074 1/20 0.59
PSMB2 P49721 1/20 0.59
GCGR P47871 1/20 0.59
MCHR1 Q99705 1/20 0.58
APP P05067 1/20 0.58
ESR1 P03372 7/20 0.57
ESR2 Q92731 7/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7452408 0.96 ESR1 (0.64) CNR1BCHECNR2ACHELTA4H
SCHEMBL11734690 0.96 LTA4H (0.63) CNR1BCHECNR2ACHELTA4H
SCHEMBL7447390 0.95 L3MBTL1 (0.69) CNR1BCHECNR2ACHELTA4H
SCHEMBL7946033 0.95 ESR1 (0.65) CNR1BCHECNR2ACHELTA4H
SCHEMBL11730136 0.94 L3MBTL1 (0.68) CNR1BCHECNR2ACHELTA4H
Hydrochloric Acid SCHEMBL6749954 0.94 ESR1 (0.66) CNR1BCHECNR2ACHELTA4H
Hydrochloric Acid SCHEMBL6748794 0.93 L3MBTL1 (0.67) CNR1BCHECNR2ACHEL3MBTL1
SCHEMBL11728245 0.90 BCHE (0.57) CNR1BCHECNR2ACHELTA4H
SCHEMBL8591606 0.86 ESR1 (0.70) CNR1ACHEESR1ESR2
SCHEMBL7946146 0.85 ESR1 (0.67) CNR1ACHELTA4HESR1ESR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6265575-B1 THROMBIN INHIBITORS ELI LILLY AND COMPANY 2001-07-24 US disclosed
US-6251921-B1 ADMINISTERING THROMBIN INHIBITING DIAMINE COMPOUND TO MAMMAL ELI LILLY AND COMPANY 2001-06-26 US disclosed
US-6025382-A Antithrombotic diamines ELI LILLY AND COMPANY (US) 2000-02-15 US disclosed
EP-0863755-A4 ANTITHROMBOTIC DIAMINES LILLY CO ELI (US) 1999-01-20 EP disclosed
EP-0863755-A1 ANTITHROMBOTIC DIAMINES ELI LILLY AND COMPANY (US) 1998-09-16 EP disclosed
WO-1997025033-A1 ANTITHROMBOTIC DIAMINES ELI LILLY AND COMPANY (US) 1997-07-17 WO disclosed