SCHEMBL7452883

SCHEMBL7452883

CN[C@H]1CCN(Cc2cccc3nc(O)ccc23)C1=O

nearest known ligand 0.36

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 2/20 0.36
HDAC8 Q9BY41 1/20 0.36
HDAC6 Q9UBN7 1/20 0.36
F10 P00742 13/20 0.34
F2 P00734 2/20 0.34
PLG P00747 2/20 0.34
PLAT P00750 2/20 0.34
PROC P04070 2/20 0.34
PRSS1 P07477 2/20 0.34
ACE P12821 1/20 0.34
XIAP P98170 1/20 0.34
HCRTR2 O43614 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7452877 0.87 HDAC1 (0.35) HDAC1HDAC8HDAC6F10F2
SCHEMBL7220633 0.86 F10 (0.42) HDAC1HDAC8HDAC6F10F2
Trifluoroacetic Acid SCHEMBL7214094 0.81 F10 (0.40) HDAC1HDAC8HDAC6F10F2
SCHEMBL7214254 0.81 TSHR (0.32) HDAC1ACEHCRTR2
SCHEMBL7214250 0.80 ELANE (0.34) HDAC1HCRTR2
SCHEMBL7454004 0.78 F10 (0.43) F10F2PLGPROC
SCHEMBL7214087 0.72 ACACB (0.42) F10F2PLGPLATPROC
SCHEMBL7937461 0.72 HDAC1 (0.56) HDAC1HDAC8HDAC6F10ACE
SCHEMBL7937458 0.72 HDAC1 (0.56) HDAC1HDAC8HDAC6F10ACE
SCHEMBL5604870 0.71 ALDH1A1 (0.49)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0944386-B1 SULFONIC ACID OR SULFONYLAMINO N-(HETEROARALKYL)-AZAHETEROCYCLYLAMIDE COMPOUNDS AVENTIS PHARMA INC (US) 2002-09-18 EP claimed
EP-0944386-B1 SULFONIC ACID OR SULFONYLAMINO N-(HETEROARALKYL)-AZAHETEROCYCLYLAMIDE COMPOUNDS AVENTIS PHARMA INC (US) 2002-09-18 EP disclosed
WO-2001039759-A2 SULFONIC ACID OR SULFONYLAMINO N-(HETEROARALKYL)-AZAHETEROCYCLYLAMIDE COMPOUNDS AVENTIS PHARMA DEUTSCHLAND GMBH (DE) 2001-06-07 WO disclosed