SCHEMBL7455076

SCHEMBL7455076

NCC(CCC(c1ccccc1)c1ccccc1)C(=O)O

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRM2 Q14416 2/20 0.54
GRM3 Q14832 2/20 0.54
HRH1 P35367 2/20 0.52
HTR2A P28223 2/20 0.50
TAAR1 Q96RJ0 1/20 0.50
EPHX2 P34913 1/20 0.47
GABBR2 O75899 1/20 0.47
GABBR1 Q9UBS5 1/20 0.47
MTNR1A P48039 1/20 0.44
MTNR1B P49286 1/20 0.44
CYP1A2 P05177 1/20 0.44
CYP2D6 P10635 1/20 0.43
SRC P12931 1/20 0.43
CNR1 P21554 1/20 0.43
CNR2 P34972 1/20 0.43
SLC1A2 P43004 1/20 0.43
SLC1A1 P43005 1/20 0.43
CHRNB2 P17787 1/20 0.42
CHRNA4 P43681 1/20 0.42
FOLH1 Q04609 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4989765 0.84 TAAR1 (0.55) GRM2GRM3HTR2ATAAR1GABBR2
SCHEMBL13917993 0.82 GRM2 (0.68) GRM2GRM3HRH1HTR2ATAAR1
SCHEMBL4993935 0.81 GABBR2 (0.49) GRM2GRM3HTR2ATAAR1GABBR2
SCHEMBL7390788 0.77 GRIK1 (0.54) CYP1A2SLC1A2SLC1A1
SCHEMBL13917992 0.74 GRIK1 (0.69) HTR2ACYP1A2FOLH1LMNAMAPK1
SCHEMBL4985838 0.74 CYP1A2 (0.55) CYP1A2SLC1A2SLC1A1FOLH1
SCHEMBL3290730 0.73 HRH1 (0.68) HRH1HTR2ATAAR1MTNR1AMTNR1B
SCHEMBL4989295 0.73 GRIK1 (0.47) CYP1A2
SCHEMBL6452470 0.73 MTNR1A (0.49) MTNR1AMTNR1BCYP1A2
SCHEMBL4738634 0.72 CYP1A2 (0.76) CYP1A2SLC1A2SLC1A1FOLH1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7501429-B2 Pyrimidine compounds as anti-ictogenic and/or anti-epileptogenic agents QUEEN'S UNIVERSITY AT KINGSTON (CA) 2009-03-10 US disclosed
US-7501429-B2 Pyrimidine compounds as anti-ictogenic and/or anti-epileptogenic agents QUEEN'S UNIVERSITY AT KINGSTON (CA) 2009-03-10 US disclosed
EP-1230260-A1 HCV NS3 PROTEASE INHIBITORS ISTITUTO DI RICERCHE DI BIOLOGIA MOLECOLARE P. ANGELETTI S.P.A. (IT) 2002-08-14 EP disclosed
WO-2001032691-A1 HCV NS3 PROTEASE INHIBITORS ISTITUTO DI RICERCHE DI BIOLOGIA MOLECOLARE P. ANGELETTI S.P.A. (IT) 2001-05-10 WO disclosed