SCHEMBL7455117

SCHEMBL7455117

C1=C(c2ccc3sccc3c2)CC2CCC1N2

nearest known ligand 0.60

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 3/20 0.46
CHRNA4 P43681 3/20 0.46
P2RY14 Q15391 1/20 0.40
DYRK1A Q13627 1/20 0.39
CA12 O43570 1/20 0.38
ENPP1 P22413 1/20 0.38
HTR6 P50406 1/20 0.36
CCNT1 O60563 1/20 0.36
CDK9 P50750 1/20 0.36
KDM1A O60341 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1023489 0.77 CHRNB2 (0.54) CHRNB2CHRNA4P2RY14CCNT1CDK9
SCHEMBL1023383 0.75 CHRNB2 (0.48) CHRNB2CHRNA4P2RY14
Hydrochloric Acid SCHEMBL1072684 0.74 CHRNB2 (0.47) CHRNB2CHRNA4P2RY14
SCHEMBL1022339 0.73 CHRNB2 (0.52) CHRNB2CHRNA4P2RY14CCNT1CDK9
SCHEMBL1022337 0.73 CHRNB2 (0.52) CHRNB2CHRNA4P2RY14CCNT1CDK9
SCHEMBL7809874 0.70 CHRNB2 (0.55) CHRNB2CHRNA4P2RY14CCNT1CDK9
SCHEMBL6993886 0.70 CHRNB2 (0.55) CHRNB2CHRNA4P2RY14CCNT1CDK9
SCHEMBL2881954 0.70 CHRNB2 (0.67) CHRNB2CHRNA4P2RY14CCNT1CDK9
SCHEMBL12093045 0.70 CHRNB2 (0.67) CHRNB2CHRNA4P2RY14CCNT1CDK9
SCHEMBL5760094 0.69 DYRK1A (0.40) DYRK1ACA12ENPP1KDM1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1242419-A1 AZABICYCLO 3.2.1]OCTANE DERIVATIVES ELI LILLY AND COMPANY (US) 2002-09-25 EP disclosed
WO-2001046187-A1 AZABICYCLO[3.2.1]OCTANE DERIVATIVES ELI LILLY AND COMPANY (US) 2001-06-28 WO disclosed