SCHEMBL7455356

SCHEMBL7455356

COC(=O)c1cc(CC2SC(=O)NC2=O)ccc1OC

nearest known ligand 0.63

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PTPN1 P18031 2/20 0.63
CA2 P00918 1/20 0.53
ALDH1A1 P00352 1/20 0.52
NPSR1 Q6W5P4 1/20 0.52
PPARG P37231 8/20 0.49
MPC2 O95563 2/20 0.49
CYP2C8 P10632 2/20 0.49
CYP2C9 P11712 2/20 0.49
MAOA P21397 2/20 0.49
CISD1 Q9NZ45 2/20 0.49
MAPT P10636 2/20 0.49
MAOB P27338 1/20 0.47
FFAR1 O14842 3/20 0.44
LMNA P02545 1/20 0.44
HPGD P15428 1/20 0.44
PPARA Q07869 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5707014 0.89 PTPN1 (0.64) PTPN1CA2ALDH1A1NPSR1PPARG
SCHEMBL6447702 0.86 ALDH1A1 (0.53) PTPN1CA2ALDH1A1NPSR1PPARG
SCHEMBL8182679 0.84 PTPN1 (0.79) PTPN1CA2ALDH1A1NPSR1PPARG
SCHEMBL13524845 0.83 PTPN1 (0.55) PTPN1CA2ALDH1A1NPSR1PPARG
SCHEMBL13847876 0.82 PTPN1 (0.54) PTPN1CA2ALDH1A1NPSR1PPARG
SCHEMBL14262660 0.82 PTPN1 (0.68) PTPN1CA2ALDH1A1NPSR1PPARG
SCHEMBL6231739 0.82 PPARA (0.55) PTPN1CA2ALDH1A1NPSR1PPARG
SCHEMBL13846691 0.81 PTPN1 (0.67) PTPN1CA2ALDH1A1NPSR1PPARG
SCHEMBL6233368 0.81 PTPN1 (0.67) PTPN1CA2ALDH1A1NPSR1PPARG
SCHEMBL6376424 0.81 POLB (0.54) PTPN1CA2ALDH1A1PPARGLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1133627-C Intermediate of N-benzyl dioxothiazolidinyl benzoyl amide derivatives, and its prepn. method ������ҩ��ʽ���� 2004-01-07 CN disclosed
CN-1336366-A Intermediate of N-benzyl dioxothiazolidinyl benzoyl amide derivatives, and its prepn. method KYORIN SEIYAKU KK (JP) 2002-02-20 CN disclosed
EP-0846693-B1 N-BENZYLDIOXOTHIAZOLIDYLBENZAMIDE DERIVATIVES AND PROCESS FOR PRODUCING THE SAME KYORIN SEIYAKU KK (JP) 2002-01-23 EP disclosed
CN-1069901-C N-benzyldioxothiazolidylbenzamide derivatives and process for producing the same KYORIN SEIYAKU KK (JP) 2001-08-22 CN disclosed
US-6147101-A TREATING HYPERGLYCEMIA KYORIN PHARMACEUTICAL CO., LTD. (JP) 2000-11-14 US disclosed
US-6030990-A ANTIDIABETIC AND -LIPEMIC AGENTS; PARTICULARLY FOR NON-INSULIN DEPENDENT DIABETES MELLITUS, A BLOOD SUGAR-LOWERING DRUG THAT IMPROVES THE INSULIN RESISTANCE AND HAS HIGH SAFETY AND EFFICIENCY KYORIN PHARMACEUTICAL CO., LTD. (JP) 2000-02-29 US disclosed
US-6001862-A ADMINISTERING TO A PATIENT SUFFERING FROM NON-INSULIN DEPENDENT DIABETES MELLITUS A N-BENZYLDIOXOTHIAZOLIDYLBENZAMIDE COMPOUND KYORIN PHARAMEUTICALS CO., LTD. (JP) 1999-12-14 US disclosed
CN-1186489-A N-benzyldioxothiazolidylbenzamide derivatives and process for producing the same KYORIN SEIYAKU KK (JP) 1998-07-01 CN disclosed
EP-0846693-A1 N-BENZYLDIOXOTHIAZOLIDYLBENZAMIDE DERIVATIVES AND PROCESS FOR PRODUCING THE SAME KYORIN PHARMACEUTICAL CO., LTD. (JP) 1998-06-10 EP disclosed