SCHEMBL7455757

SCHEMBL7455757

COC(=O)C(N)(C#CCc1ccccc1)S(=O)(=O)c1sccc1S(=O)(=O)c1ccccc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 1/20 0.39
KDM4E B2RXH2 2/20 0.39
ALDH1A1 P00352 2/20 0.35
GAA P10253 1/20 0.35
PKM P14618 1/20 0.35
HPGD P15428 1/20 0.35
MMP1 P03956 5/20 0.35
MMP13 P45452 5/20 0.35
MMP9 P14780 3/20 0.35
PTPRB P23467 2/20 0.34
PTPN2 P17706 1/20 0.34
PTPN1 P18031 1/20 0.34
PTPRA P18433 1/20 0.34
MMP2 P08253 3/20 0.33
MMP3 P08254 2/20 0.33
LMNA P02545 1/20 0.33
KMT2A Q03164 1/20 0.33
CA4 P22748 2/20 0.32
CNR1 P21554 1/20 0.32
ABCC9 O60706 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7455316 0.75 MMP13 (0.40) ALDH1A1MMP1MMP13MMP9PTPRB
SCHEMBL7450820 0.72 NPSR1 (0.43) NPSR1KDM4EALDH1A1MMP13MMP9
SCHEMBL3283084 0.65 NPSR1 (0.57) NPSR1KDM4EALDH1A1GAAKMT2A
SCHEMBL4250028 0.64 NPSR1 (0.60) NPSR1KDM4EALDH1A1GAAMMP1
SCHEMBL27853854 0.63 KCNN4 (0.46) KDM4EALDH1A1GAAPKMHPGD
Hydrochloric Acid SCHEMBL27583303 0.63 NPSR1 (0.58) NPSR1KDM4EALDH1A1GAAMMP1
SCHEMBL7512000 0.62 POLB (0.42) ALDH1A1HPGDMMP1MMP13MMP9
SCHEMBL787867 0.61 NPSR1 (0.56) NPSR1KDM4EALDH1A1GAAMMP1
SCHEMBL7679168 0.61 TAAR1 (0.48) LMNATP53
SCHEMBL1466372 0.60 FFAR1 (0.42) ALDH1A1LMNAKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1165501-A1 ALKENYL- AND ALKYNYL-CONTAINING METALLOPROTEASE INHIBITORS THE PROCTER & GAMBLE COMPANY (US) 2002-01-02 EP disclosed
US-6197770-B1 ENZYME INHIBITORS; ANTIARTHRITIC AGENTS; BONE DISORDERS THE PROCTER & GAMBLE CO. 2001-03-06 US disclosed
WO-2000051975-A1 ALKENYL- AND ALKYNYL-CONTAINING METALLOPROTEASE INHIBITORS THE PROCTER & GAMBLE COMPANY (US) 2000-09-08 WO disclosed