SCHEMBL7456409

SCHEMBL7456409

CCOP(=O)(CCCn1c(=O)[nH]c2nc(CC)n(C)c2c1=O)OCC

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2B P29275 9/20 0.34
ADORA3 P0DMS8 4/20 0.34
ADORA2A P29274 3/20 0.34
PDE4A P27815 2/20 0.34
PDE4B Q07343 2/20 0.34
PDE4C Q08493 2/20 0.34
PDE4D Q08499 2/20 0.34
USP2 O75604 3/20 0.32
POLB P06746 3/20 0.32
MEN1 O00255 2/20 0.32
KMT2A Q03164 2/20 0.32
KEAP1 Q14145 2/20 0.32
NFE2L2 Q16236 2/20 0.32
SMN1; SMN2 Q16637 2/20 0.32
ALDH1A1 P00352 2/20 0.32
RGS12 O14924 1/20 0.32
NPC1 O15118 1/20 0.32
RAB9A P51151 1/20 0.32
BLM P54132 1/20 0.32
CACNA1B Q00975 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7456006 0.97 ADORA2B (0.34) ADORA2BADORA3ADORA2APDE4APDE4B
SCHEMBL8660273 0.88 ADORA2B (0.33) ADORA2BADORA3ADORA2APDE4APDE4B
SCHEMBL8657823 0.87 USP2 (0.33) ADORA2BADORA3ADORA2APDE4APDE4B
SCHEMBL10650075 0.74 MEN1 (0.35) ADORA2BADORA3ADORA2APDE4APDE4B
SCHEMBL4445212 0.70 KDM4E (0.51) ADORA2BADORA3ADORA2APDE4APDE4B
SCHEMBL3228294 0.68 ATM (0.46) POLBMEN1KMT2AALDH1A1RAB9A
SCHEMBL12152136 0.68 PDE4A (0.40) ADORA2BADORA3ADORA2APDE4APDE4B
SCHEMBL7460040 0.66 TNF (0.63) ADORA2BADORA2APDE4APDE4BPDE4C
SCHEMBL3235516 0.65 SMN1; SMN2 (0.49) USP2KMT2ASMN1; SMN2ALDH1A1HPGD
SCHEMBL8660274 0.65 CNOT7 (0.49) ADORA2BADORA3ADORA2APDE4APDE4B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0771813-B1 Alkylxanthine phosphonates and alkylxanthine phosphine oxydes and their use as medicines HOECHST AG (DE) 2002-01-16 EP disclosed
EP-0771813-A1 Alkylxanthine phosphonates and alkylxanthine phosphine oxydes and their use as medicines HOECHST AKTIENGESELLSCHAFT (DE) 1997-05-07 EP disclosed