SCHEMBL7457328

SCHEMBL7457328

Nc1ccc(N)c(-c2cc[nH]c2)c1

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHEK1 O14757 2/20 0.33
CYP3A4 P08684 3/20 0.33
CYP1A2 P05177 1/20 0.33
CYP2D6 P10635 1/20 0.33
CYP19A1 P11511 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
TDP1 Q9NUW8 4/20 0.31
ALDH1A1 P00352 3/20 0.31
NPC1 O15118 2/20 0.31
RAB9A P51151 2/20 0.31
SMN1; SMN2 Q16637 2/20 0.31
TP53 P04637 1/20 0.31
TSHR P16473 1/20 0.31
MAPK1 P28482 1/20 0.31
WEE1 P30291 1/20 0.31
CASP1 P29466 1/20 0.31
IMPDH2 P12268 1/20 0.31
MEN1 O00255 3/20 0.31
KMT2A Q03164 3/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1378148 0.81 PDE10A (0.44) CHEK1CYP3A4CYP2C9CYP2C19TDP1
SCHEMBL5705096 0.78 CASP1 (0.41) CHEK1CYP3A4CYP2C9CYP2C19TDP1
SCHEMBL7465171 0.77 ASH1L (0.32) CYP3A4CYP1A2CYP2D6CYP19A1CYP2C9
SCHEMBL26690405 0.77 CYP3A4 (0.44) CHEK1CYP3A4CYP1A2CYP2D6CYP19A1
SCHEMBL7461521 0.77 ALDH1A1 (0.41) CYP3A4CYP1A2CYP2D6CYP19A1CYP2C9
SCHEMBL7466080 0.77 GAA (0.33) CHEK1CYP3A4TDP1ALDH1A1TP53
SCHEMBL7461626 0.77 PRKCI (0.30)
SCHEMBL30867599 0.75 ALDH1A1 (0.54) CYP3A4TDP1ALDH1A1NPC1RAB9A
SCHEMBL16431200 0.75 ALDH1A1 (0.54) CYP3A4TDP1ALDH1A1NPC1RAB9A
SCHEMBL30075769 0.73 TDP1 (0.50) CYP3A4TDP1ALDH1A1NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0963982-B1 New diaminobenzene derivatives and these componends containing colouring agents WELLA AG (DE) 2002-03-13 EP claimed
US-6132475-A FOR OXIDATION DYEING OF KERATIN FIBERS; INCLUDES COUPLER AND DEVELOPER, IN WHICH THE DEVELOPER IS A SUBSTITUTED 2-(FURYL, THIENYL, PYRROLYL, OR SELENOPHENE) P-DIAMINOBENZENE DERIVATIVE OF GIVEN FORMULA; COLORFASTNESS, WASHFASTNESS WELLA AKTIENGESELLSCHAFT (DE) 2000-10-17 US claimed
EP-0963982-A2 New diaminobenzene derivatives and these componends containing colouring agents Wella Aktiengesellschaft (DE) 1999-12-15 EP claimed
EP-0963982-B1 New diaminobenzene derivatives and these componends containing colouring agents WELLA AG (DE) 2002-03-13 EP disclosed
US-6132475-A FOR OXIDATION DYEING OF KERATIN FIBERS; INCLUDES COUPLER AND DEVELOPER, IN WHICH THE DEVELOPER IS A SUBSTITUTED 2-(FURYL, THIENYL, PYRROLYL, OR SELENOPHENE) P-DIAMINOBENZENE DERIVATIVE OF GIVEN FORMULA; COLORFASTNESS, WASHFASTNESS WELLA AKTIENGESELLSCHAFT (DE) 2000-10-17 US disclosed
EP-0963982-A2 New diaminobenzene derivatives and these componends containing colouring agents Wella Aktiengesellschaft (DE) 1999-12-15 EP disclosed