SCHEMBL7458908

SCHEMBL7458908

Cc1ccc(Cc2cncnc2N2CCC(=O)CC2)cc1.O=C1CCN(c2ncncc2Cc2ccc(C(F)(F)F)cc2)CC1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RPS6KB1 P23443 2/20 0.42
KIT P10721 1/20 0.39
TP53 P04637 1/20 0.38
POLB P06746 1/20 0.38
GAA P10253 1/20 0.38
MAPT P10636 1/20 0.38
IDH1 O75874 1/20 0.37
SMO Q99835 4/20 0.36
AKT1 P31749 1/20 0.36
AKT2 P31751 1/20 0.36
AKT3 Q9Y243 1/20 0.36
KDM1A O60341 1/20 0.36
BCHE P06276 1/20 0.36
ACHE P22303 1/20 0.36
CYP1A2 P05177 2/20 0.35
CYP2C19 P33261 2/20 0.35
MEN1 O00255 1/20 0.35
CYP2C9 P11712 1/20 0.35
KMT2A Q03164 1/20 0.35
P2RX3 P56373 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7157196 0.94 RPS6KB1 (0.43) RPS6KB1KITSMOAKT1AKT2
SCHEMBL7159916 0.91 PIK3CA (0.39) KITTP53POLBMAPTAKT1
SCHEMBL7160558 0.82 PIK3CA (0.42) RPS6KB1KITTP53CYP1A2CYP2C19
SCHEMBL7160406 0.82 RPS6KB1 (0.43) RPS6KB1POLBGAAAKT1MEN1
SCHEMBL7159326 0.79 MAPK1 (0.39) RPS6KB1MAPTSMOAKT1AKT2
SCHEMBL7156878 0.79 PDE10A (0.36) RPS6KB1AKT1AKT2AKT3CYP1A2
SCHEMBL7159692 0.79 KIT (0.40) KITTP53POLBMAPTACHE
SCHEMBL7163515 0.79 RPS6KB1 (0.44) RPS6KB1POLBMAPTSMOCYP2C19
SCHEMBL5206883 0.77 DHFR (0.43) RPS6KB1SMO
SCHEMBL7159379 0.75 PIK3CA (0.36) RPS6KB1AKT1AKT2CYP1A2CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2002541245-A 2002-12-03 JP claimed
EP-1165523-A1 NEUROTROPHIC SUBSTITUTED PYRIMIDINES Krenitsky Pharmaceuticals, Inc. (US) 2002-01-02 EP claimed
WO-2000061562-A1 NEUROTROPHIC SUBSTITUTED PYRIMIDINES KRENITSKY PHARMACEUTICALS INC. (US) 2000-10-19 WO claimed