SCHEMBL7459458

SCHEMBL7459458

O=C1CC(C(=O)N(CCCN2CCC(Cc3ccccc3)CC2)c2ccccc2)CN1CCCc1ccccc1

nearest known ligand 0.64

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 3/20 0.64
OPRM1 P35372 6/20 0.51
CCR3 P51677 1/20 0.50
SIGMAR1 Q99720 1/20 0.50
HRH3 Q9Y5N1 1/20 0.47
CYP2D6 P10635 1/20 0.47
SMAD3 P84022 1/20 0.47
KDM4E B2RXH2 1/20 0.46
LMNA P02545 1/20 0.46
GAA P10253 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7458584 0.95 CCR5 (0.65) CCR5OPRM1CCR3SIGMAR1CYP2D6
SCHEMBL7456733 0.92 CCR5 (0.66) CCR5OPRM1
SCHEMBL3037256 0.91 CCR5 (0.66) CCR5OPRM1
SCHEMBL7458135 0.91 CCR5 (0.57) CCR5OPRM1
Hydrochloric Acid SCHEMBL7465772 0.90 CCR5 (0.70) CCR5OPRM1
SCHEMBL7458912 0.90 CCR5 (0.62) CCR5OPRM1CYP2D6GAA
SCHEMBL7467086 0.89 CCR5 (0.63) CCR5OPRM1CCR3
SCHEMBL3032771 0.88 CCR5 (0.62) CCR5OPRM1
SCHEMBL7465873 0.88 CCR5 (0.62) CCR5OPRM1
SCHEMBL7463797 0.88 CCR5 (0.62) CCR5OPRM1CYP2D6SMAD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1180513-A1 CYCLIC AMIDE COMPOUNDS, PROCESS FOR THE PREPARATION OF THE SAME AND USES THEREOF Takeda Chemical Industries, Ltd. (JP) 2002-02-20 EP disclosed