Bromide

Bromide

SCHEMBL7460540

CC(=O)Oc1cccc2cc(C[N+](C)(C)C)cnc12.[Br-]

nearest known ligand 0.42

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACHECHKACHRM1CHRM2CHRM3CHRM4CHRM5CHRNA1CHRNB1CHRNDCHRNECHRNGHRH2OPRM1

The experimentally established mechanism targets of Bromide. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACHE known ✓ P22303 1/20 0.39
PARP1 P09874 1/20 0.42
PDE10A Q9Y233 2/20 0.41
HPGDS O60760 2/20 0.41
KDM4E B2RXH2 3/20 0.38
L3MBTL1 Q9Y468 3/20 0.38
POLB P06746 2/20 0.38
GAA P10253 2/20 0.38
ALDH1A1 P00352 2/20 0.38
KMT2A Q03164 2/20 0.38
TDP1 Q9NUW8 2/20 0.38
MAPT P10636 1/20 0.38
APEX1 P27695 1/20 0.38
RECQL P46063 1/20 0.38
BLM P54132 1/20 0.38
LMNA P02545 4/20 0.37
SMN1; SMN2 Q16637 2/20 0.37
PTPN1 P18031 1/20 0.36
METAP2 P50579 1/20 0.36
METAP1 P53582 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7597610 0.99 PARP1 (0.43) PARP1PDE10AHPGDSACHEKDM4E
SCHEMBL7594203 0.83 PARP1 (0.45) PARP1PDE10AHPGDSKDM4EL3MBTL1
SCHEMBL27444535 0.81 PDE10A (0.43) PARP1PDE10AHPGDSACHEKDM4E
Trimethylammonium SCHEMBL7594552 0.80 PARP1 (0.42) PARP1PDE10AHPGDSKDM4EL3MBTL1
Jineol Acetate SCHEMBL8608939 0.77 ALDH1A1 (0.51) PDE10AHPGDSKDM4EL3MBTL1POLB
SCHEMBL7466188 0.77 PARP1 (0.56) PARP1PDE10AHPGDSACHEKDM4E
Bromide SCHEMBL7469974 0.77 KDM4E (0.55) PARP1KDM4EKMT2AMETAP2METAP1
Bromide SCHEMBL8838429 0.74 PARP1 (0.40) PARP1PDE10AKDM4EL3MBTL1ALDH1A1
Bromide SCHEMBL8838451 0.73 PDE10A (0.50) PARP1PDE10AKDM4EL3MBTL1POLB
SCHEMBL8838373 0.71 PDE10A (0.51) PARP1PDE10AKDM4EL3MBTL1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0747362-B1 Substituted quinoline herbicide intermediates and process BASF AG (DE) 2002-10-30 EP claimed
EP-0747362-A1 Substituted quinoline herbicide intermediates and process American Cyanamid Company (US) 1996-12-11 EP claimed
CN-1100758-C Process for preparation of [(5, 6 -dicarboxy 3 -pyridyl) methyl] ammonium halides AMERICAN CYANAMID CO (US) 2003-02-05 CN disclosed
EP-0747362-B1 Substituted quinoline herbicide intermediates and process BASF AG (DE) 2002-10-30 EP disclosed
EP-0812828-B1 Process for the preparation of (5,6-dicarboxy-3-pyridyl) methyl ammonium halides BASF AG (DE) 2002-03-13 EP disclosed
US-6002012-A Process for the preparation of [(5,6-dicarboxy-3-pyridyl) methyl] ammonium halides AMERICAN CYANAMID COMPANY (US) 1999-12-14 US disclosed
CN-1172802-A Process for preparation of [(5, 6 -dicarboxy 3 -pyridyl) methyl] ammonium halides AMERICAN CYANAMID CO (US) 1998-02-11 CN disclosed
EP-0812828-A1 Process for the preparation of (5,6-dicarboxy-3-pyridyl) methyl ammonium halides American Cyanamid Company (US) 1997-12-17 EP disclosed
US-5633380-A DEHALOGENATED, DESALTED HERBICIDES AMERICAN CYANAMID COMPANY (US) 1997-05-27 US disclosed
EP-0747362-A1 Substituted quinoline herbicide intermediates and process American Cyanamid Company (US) 1996-12-11 EP disclosed