SCHEMBL7462333

SCHEMBL7462333

O=C(O)Nc1ccc(C(=O)c2ccccc2)cc1NC(=O)CC(=O)c1cccc(Cl)c1

nearest known ligand 0.49

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ERCC5 P28715 1/20 0.49
FEN1 P39748 1/20 0.49
ALDH1A1 P00352 5/20 0.47
SMN1; SMN2 Q16637 3/20 0.47
LMNA P02545 1/20 0.47
SERPINE1 P05121 1/20 0.45
MAPT P10636 5/20 0.45
RAB9A P51151 4/20 0.45
KMT2A Q03164 4/20 0.45
NPC1 O15118 2/20 0.45
MAPK1 P28482 2/20 0.44
MEN1 O00255 3/20 0.43
POLB P06746 1/20 0.43
VNN1 O95497 1/20 0.43
TP53 P04637 1/20 0.43
THRB P10828 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5868781 0.85 MAPT (0.42) ERCC5FEN1ALDH1A1SMN1; SMN2LMNA
SCHEMBL7459390 0.83 GSK3B (0.46) LMNARAB9AKMT2AVNN1
SCHEMBL8987286 0.76 NPC1 (0.69) ERCC5FEN1ALDH1A1SMN1; SMN2LMNA
SCHEMBL27597149 0.75 SERPINE1 (0.43) ERCC5FEN1ALDH1A1SMN1; SMN2LMNA
SCHEMBL1133114 0.74 ATM (0.71) ERCC5FEN1ALDH1A1RAB9ANPC1
SCHEMBL31514279 0.74 ATM (0.71) ERCC5FEN1ALDH1A1RAB9ANPC1
SCHEMBL27615911 0.73 WNT3A (0.44) ALDH1A1SMN1; SMN2SERPINE1MAPTRAB9A
SCHEMBL27615863 0.73 RAB9A (0.46) ALDH1A1SMN1; SMN2SERPINE1MAPTRAB9A
SCHEMBL14982192 0.73 ERCC5 (0.74) ERCC5FEN1ALDH1A1SMN1; SMN2LMNA
Ammonia Solution, Strong SCHEMBL28227232 0.72 ATM (0.68) ERCC5FEN1ALDH1A1RAB9ANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1224175-A2 BENZODIAZEPINE DERIVATIVES AS METABOTROPIC GLUTAMATE RECEPTOR ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2002-07-24 EP disclosed
WO-2001029012-A2 BENZODIAZEPINE DERIVATIVES AS METABOTROPIC GLUTAMATE RECEPTOR ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2001-04-26 WO disclosed