SCHEMBL7462602

SCHEMBL7462602

COc1ccc(NC(=O)ON2CCC(c3c[nH]c4ccc(F)cc34)C2)cc1N1CCN(C)CC1

nearest known ligand 0.78

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 5/20 0.52
HTR1D P28221 5/20 0.52
HTR1B P28222 5/20 0.52
HTR1F P30939 2/20 0.52
HTR2A P28223 1/20 0.49
HTR2C P28335 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7462311 0.95 HTR1D (0.55) HTR1AHTR1DHTR1BHTR1FHTR2A
SCHEMBL7463036 0.92 HTR1A (0.50) HTR1AHTR1DHTR1BHTR1F
SCHEMBL22410939 0.88 HTR1A (0.59) HTR1AHTR1DHTR1BHTR1FHTR2A
Hydrochloric Acid SCHEMBL7460920 0.87 HTR1A (0.51) HTR1AHTR1DHTR1BHTR1F
SCHEMBL6346308 0.86 HTR1A (0.63) HTR1AHTR1DHTR1BHTR1FHTR2A
SCHEMBL7461604 0.84 HTR1A (0.61) HTR1AHTR1DHTR1BHTR1FHTR2A
SCHEMBL6348488 0.84 HTR1D (0.57) HTR1AHTR1DHTR1BHTR1F
SCHEMBL7455762 0.83 HTR1A (0.54) HTR1AHTR1DHTR1BHTR1FHTR2A
SCHEMBL7461571 0.82 HTR1A (0.51) HTR1AHTR1DHTR1BHTR1FHTR2A
SCHEMBL6356041 0.80 HTR1A (0.62) HTR1AHTR1DHTR1BHTR2AHTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1140898-B1 AMIDE AND UREA DERIVATIVES AS 5-HT REUPTAKE INHIBITORS AND AS 5-HT1B/1D LIGANDS MERCK PATENT GMBH (DE) 2002-08-28 EP disclosed
EP-1140898-A1 AMIDE AND UREA DERIVATIVES AS 5-HT REUPTAKE INHIBITORS AND AS 5-HT1B/1D LIGANDS MERCK PATENT GmbH (DE) 2001-10-10 EP disclosed
WO-2000037456-A1 AMIDE AND UREA DERIVATIVES AS 5-HT REUPTAKE INHIBITORS AND AS 5-HT1B/1D LIGANDS MERCK PATENT GMBH (DE) 2000-06-29 WO disclosed