SCHEMBL7463304

SCHEMBL7463304

CSc1sc(C2NCCN2)c2c1C(=O)CC(C)(C)C2

nearest known ligand 0.50

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
GABRG2 P18507 12/20 0.50
GABRB3 P28472 12/20 0.50
GABRA5 P31644 12/20 0.50
GABRA3 P34903 10/20 0.49
GABRA1 P14867 9/20 0.49
GABRA2 P47869 9/20 0.49
LRRK2 Q5S007 7/20 0.49
NPSR1 Q6W5P4 2/20 0.48
LMNA P02545 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7454194 0.81 GABRG2 (0.46) GABRG2GABRB3GABRA5GABRA3GABRA1
SCHEMBL7444904 0.74 GABRG2 (0.56) GABRG2GABRB3GABRA5GABRA3GABRA1
SCHEMBL4918827 0.70 GABRG2 (0.52) GABRG2GABRB3GABRA5GABRA3GABRA1
SCHEMBL4401833 0.70 NPSR1 (0.68) GABRG2GABRB3GABRA5GABRA3GABRA1
SCHEMBL7452104 0.70 NPSR1 (0.68) GABRG2GABRB3GABRA5GABRA3GABRA1
SCHEMBL7457238 0.69 NPSR1 (0.56) GABRG2GABRB3GABRA5GABRA3GABRA1
SCHEMBL7369406 0.69 GABRG2 (0.60) GABRG2GABRB3GABRA5GABRA3GABRA1
SCHEMBL4931496 0.69 NPSR1 (0.62) GABRG2GABRB3GABRA5GABRA3GABRA1
SCHEMBL7459195 0.68 NPSR1 (0.75) GABRG2GABRB3GABRA5GABRA3GABRA1
SCHEMBL7458560 0.68 NPSR1 (0.64) GABRG2GABRB3GABRA5GABRA3GABRA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0937072-B1 THIENYLCYCLOHEXANONE DERIVATIVES AS LIGANDS OF THE GABA A alpha5 RECEPTOR SUBTYPE MERCK SHARP & DOHME (GB) 2002-01-09 EP claimed