SCHEMBL7463335

SCHEMBL7463335

O=CNc1ccc2[nH]cc(C3CCNCC3)c2c1

nearest known ligand 0.67

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
APP P05067 6/20 0.67
NMT2 O60551 1/20 0.55
NMT1 P30419 1/20 0.55
HTR2C P28335 2/20 0.54
ADRB2 P07550 1/20 0.54
HTR1D P28221 9/20 0.48
HTR1B P28222 9/20 0.48
HTR1A P08908 1/20 0.48
HTR1F P30939 1/20 0.48
HTR6 P50406 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20393325 0.84 HTR1D (0.54) APPHTR1DHTR1BHTR1AHTR1F
SCHEMBL12129538 0.80 APP (1.00) APPNMT2NMT1HTR2CADRB2
SCHEMBL5357785 0.80 APP (0.64) APPNMT2NMT1HTR2CADRB2
SCHEMBL4671538 0.80 HTR1D (0.74) APPNMT2NMT1HTR2CADRB2
SCHEMBL8058252 0.79 HTR1B (0.59) HTR1DHTR1BHTR1AHTR1FHTR6
SCHEMBL8058248 0.79 HTR1B (0.59) HTR1DHTR1BHTR1AHTR1FHTR6
SCHEMBL20393394 0.77 RORC (0.64) APPHTR1DHTR1BHTR1AHTR1F
SCHEMBL12129567 0.77 APP (0.82) APPNMT2NMT1HTR2CADRB2
Phosphoric Acid SCHEMBL7867945 0.77 HTR1D (0.53) HTR1DHTR1BHTR1AHTR1F
SCHEMBL7478523 0.76 HTR1D (0.60) APPNMT2NMT1HTR2CADRB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3428160-A1 HETEROBICYCLOARYL RORC2 INHIBITORS AND METHODS OF USE THEREOF Pfizer Inc (US) 2019-01-16 EP disclosed
EP-0708102-B1 5-HT1F agonists for the treatment of migraine LILLY CO ELI (US) 2002-12-11 EP disclosed
US-5721252-A PIPERIDINYL-1H-INDOLE DERIVATIVES ELI LILLY AND COMPANY (US) 1998-02-24 US disclosed
US-5521196-A ANALGESICS USING SEROTONIN ANTAGONIST ELI LILLY AND COMPANY (US) 1996-05-28 US disclosed
EP-0708102-A1 5-HT1F agonists for the treatment of migraine ELI LILLY AND COMPANY (US) 1996-04-24 EP disclosed