SCHEMBL7463569

SCHEMBL7463569

CS(=O)(=O)OCCc1ccc(-c2ccc(F)c(Cl)c2)cc1

nearest known ligand 0.53

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 9/20 0.45
HTR2A P28223 2/20 0.43
GRM2 Q14416 1/20 0.43
PTGS1 P23219 5/20 0.40
NR1H4 Q96RI1 1/20 0.39
RPA1 P27694 1/20 0.39
NR1H2 P55055 1/20 0.37
NR1H3 Q13133 1/20 0.37
MAOB P27338 2/20 0.37
DRD2 P14416 1/20 0.37
HTR2C P28335 1/20 0.37
DRD3 P35462 1/20 0.37
HTR6 P50406 1/20 0.37
TDP2 O95551 1/20 0.36
MMP2 P08253 1/20 0.36
MMP3 P08254 1/20 0.36
ERCC1 P07992 1/20 0.36
ERCC4 Q92889 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14248769 0.88 DAO (0.41) PTGS2
SCHEMBL7456595 0.82 CHKA (0.41) PTGS2PTGS1MAOB
SCHEMBL13545900 0.81 MAOB (0.46) PTGS2MAOB
SCHEMBL15229213 0.80 KCNH2 (0.42) PTGS2PTGS1
SCHEMBL1284072 0.78 CA1 (0.43)
SCHEMBL5344844 0.77 DAO (0.40) PTGS2MAOB
SCHEMBL3258334 0.76 CA2 (0.50) DRD3
SCHEMBL1938089 0.76 CA1 (0.53) MMP3
SCHEMBL980388 0.75 CA1 (0.44) HTR2AMAOBHTR2C
SCHEMBL1431818 0.74 PNMT (0.47)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0837848-B1 4-ARYL-1-PHENYLALKYL-1,2,3,6-TETRAHYDROPYRIDINES HAVING NEUROTROPHIC AND NEUROPROTECTIVE ACTIVITY SANOFI SYNTHELABO (FR) 2002-09-11 EP disclosed
EP-1216996-A2 Method to synthesise biphenylyl derivatives SANOFI-SYNTHELABO (FR) 2002-06-26 EP disclosed
EP-0837848-A1 4-ARYL-1-PHENYLALKYL-1,2,3,6-TETRAHYDROPYRIDINES HAVING NEUROTROPHIC AND NEUROPROTECTIVE ACTIVITY SANOFI (FR) 1998-04-29 EP disclosed
WO-1997001536-A1 4-ARYL-1-PHENYLALKYL-1,2,3,6-TETRAHYDROPYRIDINES HAVING NEUROTROPHIC AND NEUROPROTECTIVE ACTIVITY SANOFI (FR) 1997-01-16 WO disclosed