SCHEMBL7464767

SCHEMBL7464767

O=C(O)C(Br)c1ccc(F)c(F)c1F

nearest known ligand 0.49

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CES2 O00748 5/20 0.49
CES1 P23141 5/20 0.49
ALDH1A1 P00352 1/20 0.35
BCHE P06276 1/20 0.32
PTGS1 P23219 1/20 0.31
PTGS2 P35354 1/20 0.31
EPHX2 P34913 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3638268 0.82 CES2 (0.50) CES2CES1BCHE
SCHEMBL8013319 0.79 CES2 (0.52) CES2CES1ALDH1A1BCHEPTGS1
SCHEMBL5084947 0.78 CES2 (0.65) CES2CES1ALDH1A1
SCHEMBL3733998 0.77 CES2 (0.42) CES2CES1EPHX2
SCHEMBL195340 0.76 CES2 (0.49) CES2CES1PTGS1PTGS2
SCHEMBL7478644 0.74 CES2 (0.50) CES2CES1ALDH1A1
SCHEMBL7466460 0.74 CES2 (0.50) CES2CES1ALDH1A1
SCHEMBL30882180 0.74 CES2 (0.50) CES2CES1ALDH1A1
SCHEMBL8127998 0.73 CES2 (0.47) CES2CES1ALDH1A1
SCHEMBL3635938 0.73 CES2 (0.47) CES2CES1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1077701-A4 ANTI-VIRAL COMPOUNDS LILLY CO ELI (US) 2002-03-20 EP disclosed
US-6358971-B1 FOR INHIBITING THE GROWTH OF A PICORNAVIRUS ELI LILLY AND COMPANY 2002-03-19 US disclosed
EP-1077701-A1 ANTI-VIRAL COMPOUNDS ELI LILLY AND COMPANY (US) 2001-02-28 EP disclosed
WO-1999059587-A1 ANTI-VIRAL COMPOUNDS ELI LILLY AND COMPANY (US) 1999-11-25 WO disclosed