SCHEMBL7465220

SCHEMBL7465220

COc1ccc2c(c1)C(=O)N(CCCCN1CC=C(c3ccccn3)CC1)C(C)=CO2

nearest known ligand 0.66

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 2/20 0.46
PPARG P37231 1/20 0.41
PPARA Q07869 1/20 0.41
DRD2 P14416 2/20 0.39
HTR1A P08908 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7470829 0.92 SIGMAR1 (0.48) SIGMAR1PPARGPPARADRD2
SCHEMBL7470561 0.91 SIGMAR1 (0.49) SIGMAR1DRD2HTR1A
SCHEMBL7466647 0.90 SIGMAR1 (0.44) SIGMAR1PPARGPPARAHTR1A
SCHEMBL7472651 0.89 SIGMAR1 (0.47) SIGMAR1DRD2HTR1A
SCHEMBL6171250 0.88 SIGMAR1 (0.52) SIGMAR1DRD2HTR1A
SCHEMBL7466677 0.88 SIGMAR1 (0.39) SIGMAR1HTR1A
SCHEMBL7472426 0.88 SIGMAR1 (0.51) SIGMAR1DRD2
SCHEMBL7472293 0.87 SIGMAR1 (0.49) SIGMAR1DRD2HTR1A
SCHEMBL7467271 0.86 SIGMAR1 (0.48) SIGMAR1PPARGPPARADRD2HTR1A
SCHEMBL7464077 0.85 DRD2 (0.42) SIGMAR1DRD2HTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0755930-B1 BENZOXAZEPINE DERIVATIVES, SALTS THEREOF, AND DRUGS CONTAINING THE SAME SUNTORY LTD (JP) 2002-07-31 EP disclosed
US-6337397-B1 A BENZOXAZEPINE DERIVATIVE FOR TREATMENT OF ANXIETY NEUROSIS, PHOBIAS, OBSESSIVE-COMPULSIVE DISORDERS, SCHIZOPHRENIA, POST-CARDIAC TRAUMA STRESS DISORDERS, DEPRESSION DISORDERS, PSYCHOSOMATIC DISORDERS AND OTHER PSYCHONEUROTIC DISORDERS, SUNTORY LIMITED (JP) 2002-01-08 US disclosed
US-6187769-B1 Benzoxazepine derivatives and their salts and medicaments containing the same SUNTORY LIMITED (JP) 2001-02-13 US disclosed
EP-0755930-A1 BENZOXAZEPINE DERIVATIVES, SALTS THEREOF, AND DRUGS CONTAINING THE SAME SUNTORY LIMITED (JP) 1997-01-29 EP disclosed