SCHEMBL7465701

SCHEMBL7465701

Nc1ncc(-c2ccc(-n3ccnc3)c(C(F)(F)F)c2)c(-c2ccncc2)n1

nearest known ligand 0.47

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 13/20 0.47
ADORA2A P29274 8/20 0.47
CYP1A2 P05177 2/20 0.43
CYP3A4 P08684 2/20 0.43
CYP2D6 P10635 2/20 0.43
CYP2C19 P33261 2/20 0.43
KMT2A Q03164 2/20 0.43
MEN1 O00255 1/20 0.43
ALDH1A1 P00352 1/20 0.43
LMNA P02545 1/20 0.43
MAPT P10636 1/20 0.43
CYP2C9 P11712 1/20 0.43
MAPK1 P28482 1/20 0.43
PMP22 Q01453 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
RPS6KA3 P51812 1/20 0.37
CDK5 Q00535 1/20 0.37
CDK5R1 Q15078 1/20 0.37
ADH5 P11766 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7535601 0.86 CYP1A2 (0.46) ADORA1ADORA2ACYP1A2CYP3A4CYP2D6
SCHEMBL7462501 0.79 ADORA1 (0.60) ADORA1ADORA2ACYP3A4CYP2D6KMT2A
SCHEMBL7463419 0.77 ADORA1 (0.59) ADORA1ADORA2ACDK5CDK5R1
SCHEMBL994454 0.71 CYP1A2 (0.62) CYP1A2CYP3A4CYP2D6CYP2C19KMT2A
SCHEMBL5449788 0.71 ADORA1 (0.87) ADORA1ADORA2AKMT2ARPS6KA3CDK5
SCHEMBL7222483 0.69 ADORA1 (0.75) ADORA1ADORA2AKMT2ARPS6KA3CDK5
SCHEMBL7210550 0.69 ADORA1 (0.75) ADORA1ADORA2AKMT2ARPS6KA3CDK5
SCHEMBL27560021 0.69 KDM4E (0.43) LMNAADH5
SCHEMBL7471062 0.68 ABL1 (0.51) ADORA1ADORA2ACYP1A2CYP3A4CYP2D6
SCHEMBL5456463 0.67 ADORA1 (0.74) ADORA1ADORA2AKMT2AMEN1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0233461-B2 4,5,6-Substituted-2-pyrimidinamines AMERICAN CYANAMID CO (US) 2002-05-29 EP disclosed