SCHEMBL7535601

SCHEMBL7535601

Nc1ncc(-c2ccc(-n3ccnc3)c(C(F)(F)F)c2)c(-c2ccccn2)n1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 3/20 0.46
CYP3A4 P08684 3/20 0.46
CYP2D6 P10635 3/20 0.46
CYP2C19 P33261 3/20 0.46
ALDH1A1 P00352 2/20 0.46
LMNA P02545 2/20 0.46
MEN1 O00255 1/20 0.46
MAPT P10636 1/20 0.46
CYP2C9 P11712 1/20 0.46
MAPK1 P28482 1/20 0.46
PMP22 Q01453 1/20 0.46
KMT2A Q03164 1/20 0.46
TDP1 Q9NUW8 1/20 0.46
ADORA1 P30542 10/20 0.42
ADORA2A P29274 6/20 0.42
ACVR1B P36896 1/20 0.39
TGFBR1 P36897 1/20 0.39
ALOX15 P16050 1/20 0.39
HSD17B10 Q99714 1/20 0.39
CLK4 Q9HAZ1 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7465701 0.86 ADORA1 (0.47) CYP1A2CYP3A4CYP2D6CYP2C19ALDH1A1
SCHEMBL7535967 0.80 MEN1 (0.48) CYP1A2CYP3A4CYP2D6LMNAMEN1
SCHEMBL7468146 0.80 DHFR (0.48) ADORA1ADORA2AACVR1BTGFBR1DHFR
SCHEMBL6824538 0.71 KDM4E (0.50) CYP1A2ALDH1A1LMNAMAPK1TDP1
SCHEMBL5450249 0.70 ADORA1 (0.70) ALDH1A1KMT2AADORA1ADORA2AALOX15
SCHEMBL7535607 0.69 SYK (0.54) CYP1A2CYP3A4CYP2D6CYP2C19ALDH1A1
SCHEMBL994454 0.69 CYP1A2 (0.62) CYP1A2CYP3A4CYP2D6CYP2C19ALDH1A1
SCHEMBL3722728 0.66 IDO1 (0.53) CYP1A2CYP3A4CYP2D6CYP2C19ALDH1A1
SCHEMBL7463419 0.66 ADORA1 (0.59) ADORA1ADORA2ADHFRCDK5CDK5R1
SCHEMBL29595684 0.66 CYP3A4 (1.00) CYP1A2CYP3A4CYP2D6CYP2C19ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0233461-B2 4,5,6-Substituted-2-pyrimidinamines AMERICAN CYANAMID CO (US) 2002-05-29 EP disclosed