SCHEMBL7465814

SCHEMBL7465814

COc1ccc(-n2nc(CCl)cc2-c2ccc(SC)cc2)cc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 1/20 0.52
CA2 P00918 1/20 0.52
CA9 Q16790 1/20 0.52
PTGS2 P35354 6/20 0.51
ALOX5 P09917 1/20 0.51
CCKAR P32238 11/20 0.50
PTGS1 P23219 3/20 0.50
RXRA P19793 1/20 0.48
RXRB P28702 1/20 0.48
RXRG P48443 1/20 0.48
CYP1A2 P05177 1/20 0.48
CYP3A4 P08684 1/20 0.48
CYP2C9 P11712 1/20 0.48
TSHR P16473 1/20 0.48
CYP2C19 P33261 1/20 0.48
THPO P40225 1/20 0.48
BLM P54132 1/20 0.48
PMP22 Q01453 1/20 0.48
HIF1A Q16665 1/20 0.48
NPSR1 Q6W5P4 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13239865 0.91 CA1 (0.59) CA1CA2CA9PTGS2ALOX5
SCHEMBL9297089 0.86 PTGS2 (0.65) CA1CA2CA9PTGS2ALOX5
SCHEMBL9205227 0.85 PTGS2 (0.51) PTGS2PTGS1RXRARXRBRXRG
SCHEMBL13239872 0.82 PTGS2 (0.62) CA1CA2CA9PTGS2ALOX5
SCHEMBL13239867 0.82 PTGS2 (0.58) CA1CA2CA9PTGS2ALOX5
SCHEMBL13239864 0.82 PTGS2 (0.58) CA1CA2CA9PTGS2ALOX5
SCHEMBL13239869 0.82 PTGS2 (0.62) CA1CA2CA9PTGS2ALOX5
SCHEMBL7461822 0.81 PTGS2 (0.53) CA1CA2CA9PTGS2PTGS1
SCHEMBL7465856 0.81 PTGS2 (0.54) CA1CA2CA9PTGS2ALOX5
SCHEMBL7465017 0.81 CA1 (0.64) CA1CA2CA9PTGS2ALOX5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0554829-B1 Pyrazole derivatives with antiinflammatory, analgesic and antithrombolic activity FUJISAWA PHARMACEUTICAL CO (JP) 2002-05-15 EP disclosed
US-5670533-A ANTIINFLAMMATORY AGENTS, ANALGESICS OR ANTIRHEUMATIC DISEASES FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1997-09-23 US disclosed
US-5550147-A ANTIINFLAMMATORY AGENTS, ANALGESICS, ANTITHROMBOTIC AGENTS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1996-08-27 US disclosed
EP-0554829-A2 Pyrazole derivatives with antiinflammatory, analgesic and antithrombolic activity FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1993-08-11 EP disclosed