SCHEMBL7465017

SCHEMBL7465017

COc1ccc(-n2nc(CCl)cc2-c2ccc(S(C)(=O)=O)cc2)cc1

nearest known ligand 0.64

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CA1 P00915 2/20 0.64
CA2 P00918 2/20 0.64
CA9 Q16790 2/20 0.64
PTGS2 P35354 15/20 0.64
PTGS1 P23219 9/20 0.64
ALOX5 P09917 2/20 0.55
CHRNA7 P36544 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13239865 0.89 CA1 (0.59) CA1CA2CA9PTGS2PTGS1
SCHEMBL3863035 0.88 CA1 (0.81) CA1CA2CA9PTGS2PTGS1
SCHEMBL3872673 0.88 CA1 (0.64) CA1CA2CA9PTGS2PTGS1
SCHEMBL9209865 0.86 PTGS2 (0.67) PTGS2PTGS1ALOX5
SCHEMBL7872946 0.84 PTGS2 (0.62) CA1CA2CA9PTGS2PTGS1
SCHEMBL9297089 0.84 PTGS2 (0.65) CA1CA2CA9PTGS2PTGS1
SCHEMBL8421888 0.83 PTGS2 (0.71) CA1CA2CA9PTGS2PTGS1
SCHEMBL7468149 0.82 PTGS2 (0.66) CA1CA2CA9PTGS2PTGS1
SCHEMBL3867032 0.81 CA1 (0.61) CA1CA2CA9PTGS2PTGS1
SCHEMBL7465814 0.81 CA1 (0.52) CA1CA2CA9PTGS2PTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0554829-B1 Pyrazole derivatives with antiinflammatory, analgesic and antithrombolic activity FUJISAWA PHARMACEUTICAL CO (JP) 2002-05-15 EP disclosed
US-5670533-A ANTIINFLAMMATORY AGENTS, ANALGESICS OR ANTIRHEUMATIC DISEASES FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1997-09-23 US disclosed
EP-0554829-A2 Pyrazole derivatives with antiinflammatory, analgesic and antithrombolic activity FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1993-08-11 EP disclosed