SCHEMBL7465838

SCHEMBL7465838

O=C(O)C(Br)c1cc(F)c(F)cc1F

nearest known ligand 0.40

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 3/20 0.33
PTGS2 P35354 3/20 0.33
SLC1A3 P43003 1/20 0.33
SLC1A2 P43004 1/20 0.33
SLC1A1 P43005 1/20 0.33
ALDH1A1 P00352 1/20 0.32
THRB P10828 1/20 0.32
RECQL P46063 1/20 0.32
CES2 O00748 3/20 0.31
CES1 P23141 3/20 0.31
CA1 P00915 2/20 0.31
CA2 P00918 2/20 0.31
CA4 P22748 2/20 0.31
EIF4A3 P38919 1/20 0.31
CYP2C19 P33261 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7474529 0.81 DGAT1 (0.33) CES2CES1CA1CA2CA4
SCHEMBL30882180 0.78 CES2 (0.50) ALDH1A1RECQLCES2CES1CA1
SCHEMBL7466460 0.78 CES2 (0.50) ALDH1A1CES2CES1CYP2C19
SCHEMBL7478644 0.78 CES2 (0.50) ALDH1A1RECQLCES2CES1CA1
SCHEMBL6902621 0.77 SRC (0.36) PTGS1PTGS2SLC1A3SLC1A2SLC1A1
SCHEMBL5085546 0.76 CES2 (0.39) PTGS1PTGS2SLC1A3SLC1A2SLC1A1
SCHEMBL29009873 0.76 SLC1A3 (0.38) PTGS1PTGS2SLC1A3SLC1A2SLC1A1
SCHEMBL5085545 0.76 CES2 (0.39) PTGS1PTGS2SLC1A3SLC1A2SLC1A1
SCHEMBL29653910 0.76 CES2 (0.39) PTGS1PTGS2SLC1A3SLC1A2SLC1A1
SCHEMBL3735712 0.75 PTGS1 (0.33) PTGS1PTGS2CA1CA2CA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1077701-A4 ANTI-VIRAL COMPOUNDS LILLY CO ELI (US) 2002-03-20 EP disclosed
US-6358971-B1 FOR INHIBITING THE GROWTH OF A PICORNAVIRUS ELI LILLY AND COMPANY 2002-03-19 US disclosed
EP-1077701-A1 ANTI-VIRAL COMPOUNDS ELI LILLY AND COMPANY (US) 2001-02-28 EP disclosed
WO-1999059587-A1 ANTI-VIRAL COMPOUNDS ELI LILLY AND COMPANY (US) 1999-11-25 WO disclosed