SCHEMBL7466403

SCHEMBL7466403

O=c1[nH]c2cc(F)ccc2c(=O)n1S(=O)(=O)c1ccc(Cl)cc1

nearest known ligand 0.81

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CMA1 P23946 1/20 0.81
FEN1 P39748 3/20 0.51
CA9 Q16790 5/20 0.46
CA12 O43570 5/20 0.46
CA1 P00915 4/20 0.46
CA2 P00918 4/20 0.46
PTGDR Q13258 1/20 0.42
PTGDR2 Q9Y5Y4 1/20 0.42
PARP1 P09874 1/20 0.40
MIF P14174 1/20 0.39
HTR6 P50406 1/20 0.38
PSEN1 P49768 1/20 0.38
PSEN2 P49810 1/20 0.38
APH1B Q8WW43 1/20 0.38
NCSTN Q92542 1/20 0.38
APH1A Q96BI3 1/20 0.38
PSENEN Q9NZ42 1/20 0.38
CYP19A1 P11511 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7466207 0.92 CMA1 (0.85) CMA1FEN1CA9CA12CA1
SCHEMBL7461813 0.90 CMA1 (0.68) CMA1FEN1CA9CA12CA1
SCHEMBL7463672 0.89 CMA1 (1.00) CMA1FEN1CA9CA12CA1
SCHEMBL7472683 0.85 CMA1 (0.81) CMA1FEN1CA9CA12CA1
SCHEMBL3775614 0.82 CMA1 (0.85) CMA1CA9CA12CA1CA2
SCHEMBL7465666 0.82 CMA1 (0.85) CMA1CA9CA12CA1CA2
SCHEMBL3788201 0.82 CMA1 (0.85) CMA1FEN1CA9CA12CA1
SCHEMBL7464965 0.82 CMA1 (0.85) CMA1FEN1CA9CA12CA1
SCHEMBL7467623 0.81 CMA1 (0.75) CMA1CA9CA12CA1CA2
SCHEMBL7460750 0.81 CMA1 (0.75) CMA1CA9CA12CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0795548-B1 QUINAZOLINE DERIVATIVES AND USE THEREOF SUNTORY LTD (JP) 2002-07-03 EP disclosed
US-5814631-A CHYMASE INHIBITOR, CARDIVASCULAR SUNTORY LIMITED (JP) 1998-09-29 US disclosed
EP-0795548-A1 QUINAZOLINE DERIVATIVES AND USE THEREOF SUNTORY LIMITED (JP) 1997-09-17 EP disclosed