SCHEMBL7466664

SCHEMBL7466664

COc1ccc(N2CCC(C)CC2)cc1.NCC1COc2ccccc2O1

nearest known ligand 0.66

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ADRA1D P25100 5/20 0.66
ADRA1A P35348 5/20 0.66
ADRA1B P35368 5/20 0.66
GAA P10253 3/20 0.53
SMN1; SMN2 Q16637 1/20 0.53
ALDH1A1 P00352 2/20 0.45
ADRA2A P08913 1/20 0.45
ADRA2B P18089 1/20 0.45
ADRA2C P18825 1/20 0.45
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44
POLB P06746 2/20 0.43
MAPK1 P28482 1/20 0.43
PKM P14618 1/20 0.43
CYP3A4 P08684 1/20 0.42
CYP2C9 P11712 1/20 0.42
CYP2C19 P33261 1/20 0.42
MAPT P10636 1/20 0.41
KDM4E B2RXH2 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8127003 0.99 ADRA1D (0.65) ADRA1DADRA1AADRA1BGAASMN1; SMN2
SCHEMBL7464235 0.89 ADRA1D (0.67) ADRA1DADRA1AADRA1BGAASMN1; SMN2
SCHEMBL7471577 0.89 ADRA1D (0.60) ADRA1DADRA1AADRA1BADRA2AADRA2B
Hydrochloric Acid SCHEMBL8118060 0.89 ADRA1D (0.66) ADRA1DADRA1AADRA1BGAASMN1; SMN2
Hydrochloric Acid SCHEMBL8124829 0.88 ADRA1D (0.59) ADRA1DADRA1AADRA1BADRA2AADRA2B
SCHEMBL7466853 0.83 ADRA1D (0.66) ADRA1DADRA1AADRA1BALDH1A1ADRA2A
Hydrochloric Acid SCHEMBL8117955 0.83 ADRA1D (0.64) ADRA1DADRA1AADRA1BALDH1A1ADRA2A
SCHEMBL7473732 0.80 ADRA1D (0.61) ADRA1DADRA1AADRA1BGAAALDH1A1
SCHEMBL7466659 0.80 ADRA1D (1.00) ADRA1DADRA1AADRA1BGAASMN1; SMN2
Hydrochloric Acid SCHEMBL8127001 0.79 ADRA1D (0.98) ADRA1DADRA1AADRA1BGAASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1198234-A2 BICYCLIC AROMATIC COMPOUNDS FOR TREATING DRUG ADDICTION Knoll GmbH (DE) 2002-04-24 EP claimed
WO-2001002391-A2 BICYCLIC AROMATIC COMPOUNDS FOR TREATING DRUG ADDICTION KNOLL GMBH (DE) 2001-01-11 WO claimed
EP-0717739-B1 1,4-Benzodioxane derivatives having affinity for D2 receptors and utility in the treatment of psychoses KNOLL AG (DE) 2000-03-29 EP claimed
EP-0717739-A1 BICYCLIC AROMATIC COMPOUNDS AS THERAPEUTIC AGENTS Knoll AG (DE) 1996-06-26 EP claimed
WO-1995007274-A1 BICYCLIC AROMATIC COMPOUNDS AS THERAPEUTIC AGENTS KNOLL AG (DE) 1995-03-16 WO claimed
EP-1198234-A2 BICYCLIC AROMATIC COMPOUNDS FOR TREATING DRUG ADDICTION Knoll GmbH (DE) 2002-04-24 EP disclosed
WO-2001002391-A2 BICYCLIC AROMATIC COMPOUNDS FOR TREATING DRUG ADDICTION KNOLL GMBH (DE) 2001-01-11 WO disclosed
EP-0717739-B1 1,4-Benzodioxane derivatives having affinity for D2 receptors and utility in the treatment of psychoses KNOLL AG (DE) 2000-03-29 EP disclosed