SCHEMBL7473732

SCHEMBL7473732

CC1CCN(c2ccccc2Cl)CC1.NCC1COc2ccccc2O1

nearest known ligand 0.61

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ADRA1D P25100 8/20 0.61
ADRA1A P35348 8/20 0.61
ADRA1B P35368 8/20 0.61
GAA P10253 2/20 0.47
ADRA2A P08913 2/20 0.46
ADRA2B P18089 2/20 0.46
ADRA2C P18825 2/20 0.46
MEN1 O00255 1/20 0.45
USP2 O75604 1/20 0.45
KMT2A Q03164 1/20 0.45
SCN1A P35498 1/20 0.43
SCN2A Q99250 1/20 0.43
SCN3A Q9NY46 1/20 0.43
HTR1A P08908 1/20 0.43
SIGMAR1 Q99720 1/20 0.43
ALDH1A1 P00352 1/20 0.42
HTT P42858 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8131925 0.99 ADRA1D (0.60) ADRA1DADRA1AADRA1BGAAADRA2A
SCHEMBL7475295 0.86 ADRA2B (0.48) ADRA1DADRA1AADRA1BADRA2AADRA2B
SCHEMBL7471577 0.85 ADRA1D (0.60) ADRA1DADRA1AADRA1BADRA2AADRA2B
SCHEMBL7466853 0.85 ADRA1D (0.66) ADRA1DADRA1AADRA1BADRA2AADRA2B
Hydrochloric Acid SCHEMBL8124829 0.84 ADRA1D (0.59) ADRA1DADRA1AADRA1BADRA2AADRA2B
SCHEMBL7468775 0.84 ADRA1D (0.64) ADRA1DADRA1AADRA1BHTR1AALDH1A1
Hydrochloric Acid SCHEMBL8117955 0.84 ADRA1D (0.64) ADRA1DADRA1AADRA1BADRA2AADRA2B
Hydrochloric Acid SCHEMBL8126599 0.83 ADRA1D (0.63) ADRA1DADRA1AADRA1BHTR1AALDH1A1
SCHEMBL7469733 0.82 ADRA1D (0.58) ADRA1DADRA1AADRA1BGAAADRA2A
Hydrochloric Acid SCHEMBL8125398 0.81 ADRA1D (0.57) ADRA1DADRA1AADRA1BGAAADRA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1198234-A2 BICYCLIC AROMATIC COMPOUNDS FOR TREATING DRUG ADDICTION Knoll GmbH (DE) 2002-04-24 EP claimed
WO-2001002391-A2 BICYCLIC AROMATIC COMPOUNDS FOR TREATING DRUG ADDICTION KNOLL GMBH (DE) 2001-01-11 WO claimed
EP-0717739-B1 1,4-Benzodioxane derivatives having affinity for D2 receptors and utility in the treatment of psychoses KNOLL AG (DE) 2000-03-29 EP claimed
EP-0717739-A1 BICYCLIC AROMATIC COMPOUNDS AS THERAPEUTIC AGENTS Knoll AG (DE) 1996-06-26 EP claimed
WO-1995007274-A1 BICYCLIC AROMATIC COMPOUNDS AS THERAPEUTIC AGENTS KNOLL AG (DE) 1995-03-16 WO claimed
EP-1198234-A2 BICYCLIC AROMATIC COMPOUNDS FOR TREATING DRUG ADDICTION Knoll GmbH (DE) 2002-04-24 EP disclosed
WO-2001002391-A2 BICYCLIC AROMATIC COMPOUNDS FOR TREATING DRUG ADDICTION KNOLL GMBH (DE) 2001-01-11 WO disclosed
EP-0717739-B1 1,4-Benzodioxane derivatives having affinity for D2 receptors and utility in the treatment of psychoses KNOLL AG (DE) 2000-03-29 EP disclosed