SCHEMBL7466903

SCHEMBL7466903

COCCOCOc1ccccc1C#N

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AR P10275 2/20 0.46
KDM4E B2RXH2 2/20 0.46
ALDH1A1 P00352 4/20 0.46
HPGD P15428 1/20 0.46
TSHR P16473 1/20 0.46
GAA P10253 2/20 0.45
POLB P06746 1/20 0.45
NPC1 O15118 3/20 0.45
RAB9A P51151 3/20 0.45
SMN1; SMN2 Q16637 3/20 0.43
MAPK1 P28482 2/20 0.43
HTR1A P08908 2/20 0.42
ADRA2A P08913 1/20 0.42
ADRA2B P18089 1/20 0.42
MAOA P21397 1/20 0.42
HTR2B P41595 1/20 0.42
USP2 O75604 1/20 0.40
TP53 P04637 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
HTR7 P34969 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29530470 0.89 KDM4E (0.57) ARKDM4EALDH1A1HPGDTSHR
SCHEMBL19527734 0.89 KDM4E (0.57) ARKDM4EALDH1A1HPGDTSHR
SCHEMBL828475 0.86 AR (0.53) ARKDM4EALDH1A1HPGDTSHR
SCHEMBL29530857 0.84 GAA (0.51) KDM4EALDH1A1HPGDTSHRGAA
SCHEMBL18587828 0.84 GAA (0.51) KDM4EALDH1A1HPGDTSHRGAA
SCHEMBL29530795 0.81 ALDH1A1 (0.51) ARKDM4EALDH1A1HPGDTSHR
SCHEMBL20607680 0.81 NPC1 (0.47) ARKDM4EALDH1A1HPGDTSHR
SCHEMBL1911338 0.81 ALDH1A1 (0.51) ARKDM4EALDH1A1HPGDTSHR
SCHEMBL30936621 0.81 ALDH1A1 (0.43) KDM4EALDH1A1HPGDTSHRGAA
SCHEMBL3297185 0.79 KDM4E (0.50) ARKDM4EALDH1A1TSHRGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1177176-A1 TRI-ARYL ACID DERIVATIVES AS PPAR RECEPTOR LIGANDS Aventis Pharma Deutschland GmbH (DE) 2002-02-06 EP disclosed
WO-2000064876-A1 TRI-ARYL ACID DERIVATIVES AS PPAR RECEPTOR LIGANDS AVENTIS PHARMA DEUTSCHLAND GMBH (DE) 2000-11-02 WO disclosed
US-5883248-A QUATERNARY AMMONIUM INTERMEDIATES ROUSSEL UCLAF (FR) 1999-03-16 US disclosed
US-5763617-A Cephalosporins ROUSSEL UCLAF (FR) 1998-06-09 US disclosed
US-5728828-A A 3-(3-CHLORO- OR IODOPROP-1-EN-1-YL),7-(2-AMINOTHIAZOL-4-YL) ((CARBOXY)(PHENYL)METHOXYIMINO)ACETAMIDO-3-CEPHEM; GRAMNEGATIVE AND -POSITIVE BACTERIA, ESP. ANTIBIOTIC-RESISTANCE STAPHYLOCOCCUS ROUSSEL UCLAF (FR) 1998-03-17 US disclosed
US-5712266-A Cephalosporins ROUSSEL UCLAF (FR) 1998-01-27 US disclosed