SCHEMBL7467199

SCHEMBL7467199

COc1[c]ccc(-c2ccc(-c3ccccc3)c(F)c2)c1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 5/20 0.38
PTGS2 P35354 3/20 0.38
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
CYP2C19 P33261 2/20 0.38
AKR1C3 P42330 2/20 0.38
AKR1C2 P52895 2/20 0.38
FABP2 P12104 1/20 0.38
TSHR P16473 1/20 0.38
AKR1C4 P17516 1/20 0.38
ADRA2B P18089 1/20 0.38
CHRM3 P20309 1/20 0.38
HTR2C P28335 1/20 0.38
DRD3 P35462 1/20 0.38
AKR1C1 Q04828 1/20 0.38
SLC22A6 Q4U2R8 1/20 0.38
LMNA P02545 1/20 0.38
CYP1A2 P05177 1/20 0.38
MAPT P10636 1/20 0.38
CYP2C9 P11712 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7468946 0.84 CYP11B1 (0.42) MEN1KMT2ACYP2C19TSHRLMNA
SCHEMBL7467261 0.84 CYP1A1 (0.41) MEN1KMT2ACYP2C19CYP1A2MAPT
SCHEMBL4905103 0.82 PTGS1 (0.38) PTGS1PTGS2MEN1KMT2ACYP2C19
SCHEMBL357701 0.82 CYP11B1 (0.40) MEN1KMT2ACYP2C19TSHRLMNA
SCHEMBL8131636 0.81 ERN1 (0.43) PTGS1PTGS2HTR2CMAPTBACE1
SCHEMBL3144056 0.81 PDGFRB (0.41) PTGS2ABCB1PGR
SCHEMBL7466430 0.79 CYP1A1 (0.44) KMT2ACYP2C19LMNACYP1A2MAPT
SCHEMBL7471853 0.79 ESR2 (0.39) MEN1KMT2ALMNAMAPTHPGD
SCHEMBL7472137 0.78 ESR2 (0.39) PTGS1PTGS2EGFR
SCHEMBL7458294 0.78 AKR1C3 (0.40) AKR1C3AKR1C2AKR1C4AKR1C1PGR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1244617-A1 SUBSTITUTED AMINOALKYLAMIDE DERIVATIVES AS ANTAGONISTS OF FOLLICLE STIMULATING HORMONE Ortho-McNeil Pharmaceutical, Inc. (US) 2002-10-02 EP claimed
WO-2001047875-A1 SUBSTITUTED AMINOALKYLAMIDE DERIVATIVES AS ANTAGONISTS OF FOLLICLE STIMULATING HORMONE ORTHO-MCNEIL PHARMACEUTICAL, INC. (US) 2001-07-05 WO claimed