SCHEMBL7471853

SCHEMBL7471853

COc1[c]ccc(-c2ccc(-c3ccccc3)cc2C)c1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR2 Q92731 1/20 0.39
SLC2A1 P11166 1/20 0.38
MAPT P10636 5/20 0.37
KDM4E B2RXH2 4/20 0.37
HPGD P15428 3/20 0.37
GAA P10253 2/20 0.37
CYP11B1 P15538 1/20 0.35
CYP11B2 P19099 1/20 0.35
EGFR P00533 1/20 0.35
ALDH1A1 P00352 2/20 0.33
MCL1 Q07820 1/20 0.33
PDE3B Q13370 1/20 0.33
PDE3A Q14432 1/20 0.33
KMT2A Q03164 3/20 0.33
LMNA P02545 2/20 0.33
L3MBTL1 Q9Y468 2/20 0.33
S1PR1 P21453 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
MEN1 O00255 2/20 0.33
NPC1 O15118 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7468946 0.87 CYP11B1 (0.42) MAPTKDM4EHPGDGAACYP11B1
SCHEMBL357701 0.86 CYP11B1 (0.40) MAPTKDM4EHPGDGAACYP11B1
SCHEMBL7466430 0.85 CYP1A1 (0.44) ESR2MAPTKDM4EHPGDGAA
SCHEMBL7472137 0.84 ESR2 (0.39) ESR2KDM4ECYP11B1CYP11B2EGFR
SCHEMBL3904470 0.83 MCL1 (0.41) MCL1BACE1
SCHEMBL7458294 0.81 AKR1C3 (0.40) CYP11B1CYP11B2S1PR1
SCHEMBL7467261 0.81 CYP1A1 (0.41) MAPTKDM4EHPGDEGFRALDH1A1
SCHEMBL7467199 0.79 PTGS1 (0.38) MAPTHPGDEGFRPDE3BPDE3A
SCHEMBL14953648 0.78 BACE1 (0.43) ESR2KDM4ECYP11B1CYP11B2ALDH1A1
SCHEMBL11466692 0.77 MCL1 (0.37) HPGDALDH1A1MCL1KMT2ANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1244617-A1 SUBSTITUTED AMINOALKYLAMIDE DERIVATIVES AS ANTAGONISTS OF FOLLICLE STIMULATING HORMONE Ortho-McNeil Pharmaceutical, Inc. (US) 2002-10-02 EP claimed
WO-2001047875-A1 SUBSTITUTED AMINOALKYLAMIDE DERIVATIVES AS ANTAGONISTS OF FOLLICLE STIMULATING HORMONE ORTHO-MCNEIL PHARMACEUTICAL, INC. (US) 2001-07-05 WO claimed