SCHEMBL7472137

SCHEMBL7472137

COc1[c]ccc(-c2ccc(-c3ccccc3)cc2Cl)c1

nearest known ligand 0.39

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ESR2 Q92731 1/20 0.39
ACLY P53396 8/20 0.39
CHEK1 O14757 2/20 0.38
ADORA2A P29274 1/20 0.36
ADORA1 P30542 1/20 0.36
CSNK2A1 P68400 2/20 0.36
KDM4E B2RXH2 1/20 0.35
ALDH1A1 P00352 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
CYP11B1 P15538 1/20 0.35
CYP11B2 P19099 1/20 0.35
PTGS2 P35354 2/20 0.35
EGFR P00533 1/20 0.34
PTGS1 P23219 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7468946 0.86 CYP11B1 (0.42) KDM4EALDH1A1L3MBTL1CYP11B1CYP11B2
SCHEMBL357701 0.84 CYP11B1 (0.40) KDM4EALDH1A1L3MBTL1CYP11B1CYP11B2
SCHEMBL7466430 0.84 CYP1A1 (0.44) ESR2CHEK1KDM4EALDH1A1L3MBTL1
SCHEMBL7471853 0.84 ESR2 (0.39) ESR2CHEK1KDM4EALDH1A1L3MBTL1
SCHEMBL9453856 0.83 ERN1 (0.43) KDM4EALDH1A1L3MBTL1PTGS2PTGS1
SCHEMBL27769458 0.82 AHR (0.44) L3MBTL1PTGS2
SCHEMBL7458294 0.80 AKR1C3 (0.40) CYP11B1CYP11B2
SCHEMBL7467261 0.79 CYP1A1 (0.41) CHEK1KDM4EALDH1A1L3MBTL1EGFR
SCHEMBL17514797 0.79 HSD11B1 (0.35)
SCHEMBL7467199 0.78 PTGS1 (0.38) PTGS2EGFRPTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1244617-A1 SUBSTITUTED AMINOALKYLAMIDE DERIVATIVES AS ANTAGONISTS OF FOLLICLE STIMULATING HORMONE Ortho-McNeil Pharmaceutical, Inc. (US) 2002-10-02 EP claimed
WO-2001047875-A1 SUBSTITUTED AMINOALKYLAMIDE DERIVATIVES AS ANTAGONISTS OF FOLLICLE STIMULATING HORMONE ORTHO-MCNEIL PHARMACEUTICAL, INC. (US) 2001-07-05 WO claimed