SCHEMBL7467771

SCHEMBL7467771

[c]1cccc(OCc2cccs2)c1-c1ccccc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.45
L3MBTL1 Q9Y468 2/20 0.41
GABRA1 P14867 1/20 0.39
GABRG2 P18507 1/20 0.39
GABRB3 P28472 1/20 0.39
GABRA5 P31644 1/20 0.39
GABRA3 P34903 1/20 0.39
GABRA2 P47869 1/20 0.39
GAA P10253 2/20 0.36
TSHR P16473 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
TRPM8 Q7Z2W7 1/20 0.35
SLC1A3 P43003 1/20 0.34
SLC1A2 P43004 1/20 0.34
SLC1A1 P43005 1/20 0.34
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2D6 P10635 1/20 0.33
CYP2C19 P33261 1/20 0.33
PDK2 Q15119 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL921513 0.78 HTT (0.48) HTTL3MBTL1GABRA1GABRG2GABRB3
SCHEMBL11382454 0.73 ALDH1A1 (0.44) L3MBTL1CYP1A2CYP2D6CYP2C19TDP1
SCHEMBL8008006 0.73 DRD1 (0.38) DRD2DRD4DRD3
SCHEMBL445160 0.72 HTT (0.41) HTTL3MBTL1GABRA1GABRG2GABRB3
SCHEMBL6616525 0.69 TDP1 (0.51) HTTL3MBTL1GABRA1GABRG2GABRB3
SCHEMBL7526397 0.69 KMT2A (0.57) HTTL3MBTL1SMN1; SMN2CYP3A4TDP1
SCHEMBL5269457 0.68 CYP1A2 (0.52) HTTL3MBTL1CYP1A2CYP3A4CYP2C19
SCHEMBL3867576 0.68 NR1I2 (0.46) HTTSMN1; SMN2CYP1A2CYP3A4CYP2C19
SCHEMBL2091154 0.68 TSHR (0.42) HTTL3MBTL1GAATSHRKMT2A
SCHEMBL1274782 0.68 CA1 (0.46) HTTL3MBTL1GAATSHRSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1244617-A1 SUBSTITUTED AMINOALKYLAMIDE DERIVATIVES AS ANTAGONISTS OF FOLLICLE STIMULATING HORMONE Ortho-McNeil Pharmaceutical, Inc. (US) 2002-10-02 EP claimed
WO-2001047875-A1 SUBSTITUTED AMINOALKYLAMIDE DERIVATIVES AS ANTAGONISTS OF FOLLICLE STIMULATING HORMONE ORTHO-MCNEIL PHARMACEUTICAL, INC. (US) 2001-07-05 WO claimed
EP-1244617-A1 SUBSTITUTED AMINOALKYLAMIDE DERIVATIVES AS ANTAGONISTS OF FOLLICLE STIMULATING HORMONE Ortho-McNeil Pharmaceutical, Inc. (US) 2002-10-02 EP disclosed
WO-2001047875-A1 SUBSTITUTED AMINOALKYLAMIDE DERIVATIVES AS ANTAGONISTS OF FOLLICLE STIMULATING HORMONE ORTHO-MCNEIL PHARMACEUTICAL, INC. (US) 2001-07-05 WO disclosed