SCHEMBL7468859

SCHEMBL7468859

c1ccc(C2CCN(CCCC(CCCNCc3cccs3)(c3ccccc3)c3ccccc3)CC2)cc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2C19 P33261 2/20 0.54
ALDH1A1 P00352 2/20 0.47
MCHR1 Q99705 1/20 0.45
KCNA3 P22001 1/20 0.43
SIGMAR1 Q99720 3/20 0.43
CARM1 Q86X55 1/20 0.43
PRMT6 Q96LA8 1/20 0.43
TSHR P16473 2/20 0.42
KMT2A Q03164 2/20 0.42
MEN1 O00255 1/20 0.42
TP53 P04637 1/20 0.42
CYP1A2 P05177 1/20 0.42
CYP3A4 P08684 1/20 0.42
CYP2D6 P10635 1/20 0.42
SLC18A3 Q16572 1/20 0.40
DRD2 P14416 1/20 0.40
CHRM2 P08172 1/20 0.38
CHRM4 P08173 1/20 0.38
CHRM5 P08912 1/20 0.38
CHRM1 P11229 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7467161 0.99 CYP2C19 (0.55) CYP2C19ALDH1A1MCHR1KCNA3SIGMAR1
SCHEMBL7465626 0.85 SIGMAR1 (0.54) CYP2C19MCHR1KCNA3SIGMAR1CARM1
Hydrochloric Acid SCHEMBL7466563 0.84 SIGMAR1 (0.53) CYP2C19MCHR1KCNA3SIGMAR1CARM1
SCHEMBL7462387 0.81 MCHR1 (0.46) CYP2C19MCHR1KCNA3SIGMAR1CARM1
Hydrochloric Acid SCHEMBL7461139 0.80 MCHR1 (0.45) CYP2C19MCHR1KCNA3SIGMAR1CARM1
SCHEMBL7459851 0.80 GLA (0.56) CYP2C19ALDH1A1MCHR1TSHRKMT2A
Hydrochloric Acid SCHEMBL7456232 0.79 GLA (0.55) CYP2C19ALDH1A1MCHR1TSHRKMT2A
SCHEMBL7466062 0.78 CHRM2 (0.61) MCHR1TSHRKMT2AMEN1TP53
Hydrochloric Acid SCHEMBL7460883 0.78 CHRM2 (0.60) MCHR1TSHRKMT2AMEN1TP53
SCHEMBL7468176 0.76 MCHR1 (0.48) MCHR1SIGMAR1DRD2CHRM2CHRM4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1219294-A1 MELANIN CONCENTRATING HORMONE ANTAGONISTS Takeda Chemical Industries, Ltd. (JP) 2002-07-03 EP claimed
EP-1219294-A1 MELANIN CONCENTRATING HORMONE ANTAGONISTS Takeda Chemical Industries, Ltd. (JP) 2002-07-03 EP disclosed