SCHEMBL7468965

SCHEMBL7468965

O=C(C=Cc1cccnc1)NCCC1CCN(Cc2ccccc2)CC1

nearest known ligand 0.81

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
BCHE P06276 17/20 0.81
ACHE P22303 17/20 0.81
MAOA P21397 5/20 0.72
MAOB P27338 4/20 0.68
CYP3A4 P08684 1/20 0.64
CYP2C9 P11712 1/20 0.64
NAMPT P43490 1/20 0.64

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7468962 1.00 BCHE (0.81) BCHEACHEMAOAMAOBCYP3A4
Hydrochloric Acid SCHEMBL4009736 0.99 BCHE (0.79) BCHEACHEMAOAMAOBCYP3A4
Hydrochloric Acid SCHEMBL4231207 0.99 BCHE (0.79) BCHEACHEMAOAMAOBCYP3A4
SCHEMBL83014 0.93 NAMPT (0.74) BCHEACHEMAOAMAOBCYP3A4
SCHEMBL83013 0.93 NAMPT (0.74) BCHEACHEMAOAMAOBCYP3A4
SCHEMBL9650895 0.90 ACHE (1.00) BCHEACHEMAOAMAOB
SCHEMBL9650908 0.90 ACHE (1.00) BCHEACHEMAOAMAOB
Hydrochloric Acid SCHEMBL9374592 0.89 BCHE (0.98) BCHEACHEMAOAMAOB
Hydrochloric Acid SCHEMBL9374603 0.89 BCHE (0.98) BCHEACHEMAOAMAOB
SCHEMBL83173 0.88 NAMPT (0.70) BCHEACHEMAOAMAOBCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0923570-B1 PYRIDYL ALKENE- AND PYRIDYL ALKINE- ACID AMIDES AS CYTOSTATICS AND IMMUNOSUPPRESSIVES FUJISAWA DEUTSCHLAND GMBH (DE) 2002-09-25 EP claimed
EP-0330026-B1 Piperidinoalkyl derivatives of carboxylic acid amides TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1994-10-05 EP claimed
US-5169856-A Cholinesterase antagonists TAKEDA CHEMICAL INDUSTRIES, INC. (JP) 1992-12-08 US claimed
EP-0330026-A1 Piperidinoalkyl derivatives of carboxylic acid amides Takeda Chemical Industries, Ltd. (JP) 1989-08-30 EP claimed