SCHEMBL7469285

SCHEMBL7469285

NS(=O)(=O)c1ccc(Nc2nccc(-c3ccccn3)n2)cc1

nearest known ligand 0.74

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
IKBKB O14920 12/20 0.74
DKK1 O94907 2/20 0.67
GSK3B P49841 2/20 0.67
MAPK8 P45983 1/20 0.61
MAPK10 P53779 1/20 0.61
CDK2 P24941 4/20 0.60
IGF1R P08069 1/20 0.60
CCNT1 O60563 2/20 0.59
CDK1 P06493 2/20 0.59
CCNB1 P14635 2/20 0.59
CDK9 P50750 2/20 0.59
CDK4 P11802 1/20 0.58
AURKA O14965 1/20 0.57
AURKB Q96GD4 1/20 0.57
CCNA2 P20248 1/20 0.57
CDK7 P50613 1/20 0.57
CCNH P51946 1/20 0.57
CCNA1 P78396 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7464681 0.86 CDK1 (0.61) IKBKBCDK2CCNT1CDK1CCNB1
SCHEMBL3519939 0.85 IKBKB (1.00) IKBKBDKK1GSK3BMAPK8MAPK10
SCHEMBL3519764 0.84 IKBKB (0.97) IKBKBDKK1GSK3BMAPK8MAPK10
SCHEMBL3521197 0.82 IKBKB (0.71) IKBKBDKK1GSK3BMAPK8MAPK10
SCHEMBL4894535 0.82 SYK (0.62) IKBKBCDK2CDK1CDK9CDK4
SCHEMBL7470857 0.81 ABL1 (0.63) IKBKBCDK2CDK1CCNB1CDK4
SCHEMBL1652316 0.81 IKBKB (0.64) IKBKBDKK1GSK3BAURKAAURKB
SCHEMBL3524651 0.81 IKBKB (0.70) IKBKBDKK1GSK3BMAPK8MAPK10
SCHEMBL3520305 0.81 IKBKB (0.70) IKBKBDKK1GSK3BMAPK8MAPK10
SCHEMBL3517977 0.81 IKBKB (0.70) IKBKBDKK1GSK3BMAPK8MAPK10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0233461-B2 4,5,6-Substituted-2-pyrimidinamines AMERICAN CYANAMID CO (US) 2002-05-29 EP disclosed