SCHEMBL7469696

SCHEMBL7469696

CC(C)S(=O)(=O)NCC(C)(C)C1CCC(=O)CC1

nearest known ligand 0.34

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
GRIA1 P42261 4/20 0.34
GRIA4 P48058 4/20 0.34
GRIA2 P42262 1/20 0.30
GRIA3 P42263 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7469496 0.74 GRIA1 (0.44) GRIA1GRIA4GRIA2GRIA3
SCHEMBL7477390 0.71 GRIA1 (0.51) GRIA1GRIA4GRIA2GRIA3
SCHEMBL112039 0.68 SLC2A1 (0.41)
SCHEMBL13154416 0.67 GRIA1 (0.50) GRIA1GRIA4GRIA2GRIA3
SCHEMBL8706325 0.66 CES2 (0.32)
SCHEMBL28982666 0.66 CES2 (0.32)
SCHEMBL12326283 0.66 CES2 (0.39)
SCHEMBL27902476 0.66 CES2 (0.32)
SCHEMBL11460960 0.65 CES2 (0.31)
SCHEMBL15489379 0.64 GRIA1 (0.46) GRIA1GRIA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0937708-B1 Sulphonamide derivatives LILLY CO ELI (US) 2002-12-18 EP disclosed
US-6362230-B1 ALZHEIMER'S DISEASE ELI LILLY AND COMPANY 2002-03-26 US disclosed
US-6174922-B1 FOR POTENTIATING GLUTAMATE RECEPTOR FUNCTION IN WARM BLOODED MAMMAL ELI LILLY AND COMPANY 2001-01-16 US disclosed
WO-1999043285-A2 SULPHONAMIDE DERIVATIVES ELI LILLY AND COMPANY (US) 1999-09-02 WO disclosed
EP-0937708-A2 sulphonamide derivatives ELI LILLY AND COMPANY (US) 1999-08-25 EP disclosed