SCHEMBL7469709

SCHEMBL7469709

CCCCCCCC#Cc1ncccn1

nearest known ligand 0.50

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 2/20 0.50
FAAH O00519 2/20 0.40
CES1 P23141 2/20 0.40
GPR84 Q9NQS5 1/20 0.40
FFAR1 O14842 1/20 0.39
FFAR4 Q5NUL3 1/20 0.39
CYSLTR2 Q9NS75 1/20 0.38
CYSLTR1 Q9Y271 1/20 0.38
MMP2 P08253 1/20 0.38
MMP12 P39900 1/20 0.38
ADORA3 P0DMS8 1/20 0.38
TLR7 Q9NYK1 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29263735 0.81 KDM4E (0.46) KCNH2TLR7
SCHEMBL9741847 0.78 KDM4E (0.47) ADORA3TLR7
SCHEMBL28075262 0.78 KCNH2 (0.41) KCNH2GPR84FFAR1FFAR4CYSLTR2
SCHEMBL28075142 0.78 KCNH2 (0.41) KCNH2GPR84FFAR1FFAR4CYSLTR2
SCHEMBL8639129 0.77 KCNH2 (0.46) KCNH2FAAHCES1
SCHEMBL15437934 0.74 KCNH2 (0.44) KCNH2FAAHCES1FFAR1FFAR4
SCHEMBL6371432 0.72 KCNH2 (0.58) KCNH2GPR84FFAR1FFAR4CYSLTR2
SCHEMBL5886568 0.72 FFAR1 (0.51) KCNH2GPR84FFAR1FFAR4MMP2
SCHEMBL29187197 0.72 FFAR1 (0.51) KCNH2GPR84FFAR1FFAR4MMP2
SCHEMBL5886652 0.71 FFAR1 (0.63) KCNH2GPR84FFAR1FFAR4MMP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0817773-B1 PYRIMIDINE COMPOUNDS QINETIQ LTD (GB) 2002-06-12 EP disclosed
US-6121448-A LIQUID CRYSTALLINE COMPOUNDS THE SECRETARY OF STATE FOR DEFENCE IN HER BRITTANIC MAJESTY'S GOVERNMENT OF THE UNITED KINGDOM OF GREAT BRITAIN AND NORTHERN IRELAND (GB) 2000-09-19 US disclosed
US-5986096-A REACTION OF HYDROGEN IODIDE WITH CHLORO-5-BROMOPYRIMIDINE THE SECRETARY OF STATE FOR DEFENCE IN HER BRITANNIC MAJESTY'S A GOVERNMENT OF THE U.K. OF GT. BRITAIN & N. IRELAND OF DEFENCE EVALUATION & RESEARCH AGENCY (GB) 1999-11-16 US disclosed
EP-0817773-A2 PYRIMIDINE COMPOUNDS THE SECRETARY OF STATE FOR DEFENCE (GB) 1998-01-14 EP disclosed
WO-1996030344-A2 PYRIMIDINE COMPOUNDS THE SECRETARY OF STATE FOR DEFENCE (GB) 1996-10-03 WO disclosed