SCHEMBL7470168

SCHEMBL7470168

CCOC(=O)c1ccc(NC2CCNCC2)nc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HCAR3 P49019 3/20 0.51
NMT2 O60551 2/20 0.51
NMT1 P30419 2/20 0.51
ALOX15 P16050 1/20 0.46
TRPV4 Q9HBA0 1/20 0.45
RAB9A P51151 3/20 0.44
KDM4E B2RXH2 1/20 0.44
NPC1 O15118 1/20 0.44
MAPT P10636 1/20 0.44
NOS2 P35228 2/20 0.44
CDK4 P11802 1/20 0.43
CDK6 Q00534 1/20 0.43
P2RY12 Q9H244 1/20 0.43
PRKAB2 O43741 1/20 0.42
PRKAG1 P54619 1/20 0.42
PRKAA2 P54646 1/20 0.42
PRKAA1 Q13131 1/20 0.42
PRKAG3 Q9UGI9 1/20 0.42
PRKAG2 Q9UGJ0 1/20 0.42
PRKAB1 Q9Y478 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1542815 0.91 HCAR3 (0.61) HCAR3ALOX15TRPV4RAB9AKDM4E
SCHEMBL4233677 0.87 HCAR3 (0.56) HCAR3KDM4ECDK4PRKAB2PRKAG1
SCHEMBL4217728 0.86 HCAR3 (0.48) HCAR3NMT2NMT1ALOX15TRPV4
SCHEMBL17830863 0.85 HDAC1 (0.44) NMT2NMT1ALOX15RAB9AMAPT
SCHEMBL12893939 0.82 RAB9A (0.57) ALOX15RAB9ANPC1MAPT
SCHEMBL4231706 0.80 P2RY12 (0.47) HCAR3TRPV4RAB9AKDM4ENPC1
SCHEMBL12277201 0.80 HCAR3 (0.79) HCAR3PRKAB2PRKAG1PRKAA2PRKAA1
Hydrochloric Acid SCHEMBL28763502 0.79 CA12 (0.47) NMT2NMT1RAB9ANPC1MAPT
Hydrochloric Acid SCHEMBL28763503 0.79 CA12 (0.47) NMT2NMT1RAB9ANPC1MAPT
SCHEMBL1938176 0.79 HCAR3 (0.59) HCAR3HRH3TDO2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1214313-A2 HETEROARYLOXY PROPANOLAMINES, PREPARATION METHOD AND PHARMACEUTICAL COMPOSITIONS CONTAINING SAME SANOFI-SYNTHELABO (FR) 2002-06-19 EP disclosed
WO-2001017989-A2 HETEROARYLOXYPROPANOLAMINES AS BETA3-ADRENERGIC RECEPTOR AGONISTS SANOFI-SYNTHELABO (FR) 2001-03-15 WO disclosed